Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50017411
TargetTrace amine-associated receptor 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM29135(CHEMBL11608 | cid_5610 | tyramine | p-Tyramine)
Affinity DataEC50:  990nMAssay Description:Agonist activity at human TAAR1 stably expressed in HEK293 cells incubated for 30 mins by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTrace amine-associated receptor 1(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM29135(CHEMBL11608 | cid_5610 | tyramine | p-Tyramine)
Affinity DataEC50:  30nMAssay Description:Agonist activity at rat TAAR1 stably expressed in HEK293 cells incubated for 30 mins by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetTrace amine-associated receptor 1(Mouse)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM29135(CHEMBL11608 | cid_5610 | tyramine | p-Tyramine)
Affinity DataEC50:  280nMAssay Description:Agonist activity at mouse TAAR1 stably expressed in HEK293 cells incubated for 30 mins by cAMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSigma non-opioid intracellular receptor 1(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50601684(CHEMBL5169925)
Affinity DataKd:  1.24E+4nMAssay Description:Binding affinity to sigma 1 receptor (unknown origin) assessed as dissociation constant by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSigma intracellular receptor 2(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50601684(CHEMBL5169925)
Affinity DataKd:  6.60E+3nMAssay Description:Binding affinity to sigma 2 receptor (unknown origin) assessed as dissociation constant by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed