Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50015017
TargetCyclin-dependent kinase 9(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM187120(US9670161, 1 5-Fluoro-4-(4-fluoro-2-methoxyphenyl)...)
Affinity DataKd:  1.30nMAssay Description:Inhibition of CDK9 (unknown origin) assessed as dissociation constant by DiscoveryX assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 alpha(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM187120(US9670161, 1 5-Fluoro-4-(4-fluoro-2-methoxyphenyl)...)
Affinity DataKd:  7.40nMAssay Description:Inhibition of GSK3 alpha (unknown origin) assessed as dissociation constant by DiscoveryX assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetInterleukin-1 receptor-associated kinase 1(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM187120(US9670161, 1 5-Fluoro-4-(4-fluoro-2-methoxyphenyl)...)
Affinity DataKd:  61nMAssay Description:Inhibition of IRAK1 (unknown origin) assessed as dissociation constant by DiscoveryX assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetCyclin-dependent kinase 9(Human)
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50528809(CHEMBL4589249)
Affinity DataIC50: 6nMAssay Description:Inhibition of CDK9 (unknown origin) in high presence of high ATP incubated for 25 min by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed