Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50013977
TargetMuscarinic acetylcholine receptor M3(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50370682(SOLIFENACIN)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at muscarinic M3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50571307(CHEMBL566204)
Affinity DataIC50: 733nMAssay Description:Antagonist activity at muscarinic M3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50571305(CHEMBL4857445)
Affinity DataIC50: 1.48E+3nMAssay Description:Antagonist activity at muscarinic M3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50571303(CHEMBL4875543)
Affinity DataIC50: 9.40E+3nMAssay Description:Antagonist activity at muscarinic M3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50571304(CHEMBL4859485)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at muscarinic M3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50571308(CHEMBL4855033)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at muscarinic M3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50571306(CHEMBL4850216)
Affinity DataIC50: 1.70E+4nMAssay Description:Antagonist activity at muscarinic M3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M3(Human)
Arkuda Therapeutics

Curated by ChEMBL
LigandPNGBDBM50571302(CHEMBL4873492)
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at muscarinic M3 receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed