Compile Data Set for Download or QSAR
Report error Found 21 Enz. Inhib. hit(s) with all data for entry = 50018647
TargetCyclin-dependent kinase 2(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443288(CHEMBL5273636)
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of human CDK2 at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCyclin-dependent kinase 2(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50443287(CHEMBL5275667)
Affinity DataIC50: 2.09E+3nMAssay Description:Inhibition of human CDK2 at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCalcitonin gene-related peptide 1(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610723(CHEMBL5285133)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of CGRP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610721(CHEMBL5271736)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of GPR119 (unknown origin) at 10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] B(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610715(CHEMBL5283462)
Affinity DataIC50: 2.45E+4nMAssay Description:Inhibition of MAO-B (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTyrosinase(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610709(CHEMBL5274281)
Affinity DataIC50: 2.79E+4nMAssay Description:Inhibition of tyrosinase (unknown origin) incubated for 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetTyrosinase(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610708(CHEMBL5282145)
Affinity DataIC50: 3.08E+4nMAssay Description:Inhibition of tyrosinase (unknown origin) incubated for 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetPurine nucleoside phosphorylase(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610707(CHEMBL5279874)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of PNP (unknown origin) expressed in Escherichia coliMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610711(CHEMBL5285907)
Affinity DataIC50: 4.81E+4nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCalcitonin gene-related peptide 1(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610721(CHEMBL5271736)
Affinity DataIC50: 5.12E+4nMAssay Description:Inhibition of CGRP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCalcitonin gene-related peptide 1(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610722(CHEMBL5271974)
Affinity DataIC50: 5.22E+4nMAssay Description:Inhibition of CGRP (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610710(CHEMBL5280972)
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610712(CHEMBL5284943)
Affinity DataIC50: 6.11E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610713(CHEMBL5273757)
Affinity DataIC50: 6.36E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetDipeptidyl peptidase 4(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610714(CHEMBL5285955)
Affinity DataIC50: 6.20E+5nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCorticoliberin(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610720(CHEMBL5286255)
Affinity DataKi:  0.700nMAssay Description:Binding affinity to CRF (unknown origin) receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCorticoliberin(Rat)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610716(CHEMBL5279390)
Affinity DataKi:  1nMAssay Description:Binding affinity to rat CRF receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCorticoliberin(Rat)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610717(CHEMBL5279909)
Affinity DataKi:  1.40nMAssay Description:Binding affinity to rat CRF receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50084875(DMP696 | [8-(2,4-dichloro-phenyl)-2,7-dimethyl-pyr...)
Affinity DataKi:  1.70nMAssay Description:Binding affinity to human CRF1 receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCorticoliberin(Rat)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610718(CHEMBL5290774)
Affinity DataKi:  2nMAssay Description:Binding affinity to rat CRF receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCorticoliberin(Rat)
Mazandaran University of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50610719(CHEMBL5291384)
Affinity DataKi:  2.60nMAssay Description:Binding affinity to rat CRF receptor assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed