Compile Data Set for Download or QSAR
Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 50018644
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610595(CHEMBL5279688)
Affinity DataIC50: 4nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610596(CHEMBL5289748)
Affinity DataIC50: 9nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610597(CHEMBL5288443)
Affinity DataIC50: 11nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610626(CHEMBL5277076)
Affinity DataIC50: 13nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610630(CHEMBL5266973)
Affinity DataIC50: 13nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610631(CHEMBL5281426)
Affinity DataIC50: 13nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610633(CHEMBL5288558)
Affinity DataIC50: 13nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610628(CHEMBL5273235)
Affinity DataIC50: 14nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610632(CHEMBL5267483)
Affinity DataIC50: 18nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610627(CHEMBL5278419)
Affinity DataIC50: 22nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610598(CHEMBL5266226)
Affinity DataIC50: 24nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610641(CHEMBL5290700)
Affinity DataIC50: 26nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610642(CHEMBL5267861)
Affinity DataIC50: 28nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610635(CHEMBL5282591)
Affinity DataIC50: 30nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610636(CHEMBL5277727)
Affinity DataIC50: 30nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610643(CHEMBL5267825)
Affinity DataIC50: 32nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610644(CHEMBL5284009)
Affinity DataIC50: 41nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610648(CHEMBL5270164)
Affinity DataIC50: 45nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610634(CHEMBL5285290)
Affinity DataIC50: 46nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610621(CHEMBL5283819)
Affinity DataIC50: 55nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610622(CHEMBL5286156)
Affinity DataIC50: 58nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610620(CHEMBL5287783)
Affinity DataIC50: 58nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610599(CHEMBL5275972)
Affinity DataIC50: 64nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610640(CHEMBL5284083)
Affinity DataIC50: 69nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610645(CHEMBL5267975)
Affinity DataIC50: 77nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610619(CHEMBL5286583)
Affinity DataIC50: 80nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610629(CHEMBL5282157)
Affinity DataIC50: 82nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610624(CHEMBL5283943)
Affinity DataIC50: 110nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610625(CHEMBL5280487)
Affinity DataIC50: 110nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610618(CHEMBL5280767)
Affinity DataIC50: 120nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610647(CHEMBL5283488)
Affinity DataIC50: 150nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610623(CHEMBL5272801)
Affinity DataIC50: 190nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610638(CHEMBL5267026)
Affinity DataIC50: 210nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610646(CHEMBL5284824)
Affinity DataIC50: 660nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610616(CHEMBL5271159)
Affinity DataIC50: 950nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610637(CHEMBL5281092)
Affinity DataIC50: 1.98E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610612(CHEMBL5274226)
Affinity DataIC50: 2.95E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM77502(cid_1239093 | SMR000211759 | MLS000587794 | 4-Meth...)
Affinity DataIC50: 3.93E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610609(CHEMBL5287181)
Affinity DataIC50: 4.10E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610608(CHEMBL5268772)
Affinity DataIC50: 5.67E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610601(CHEMBL5276856)
Affinity DataIC50: 6.83E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM57512(4-fluoranyl-N-[4-(6-methyl-1,3-benzothiazol-2-yl)p...)
Affinity DataIC50: 8.88E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610605(CHEMBL5285562)
Affinity DataIC50: 9.43E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610604(CHEMBL5272874)
Affinity DataIC50: 1.25E+4nMAssay Description:Inverse agonist activity at human GAL4-fused RORgamma LBD (262 to 507 residues) transfected in HEK293T cell measured after 24 hrs by dual luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-alpha(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610596(CHEMBL5289748)
Affinity DataIC50: 2.00E+4nMAssay Description:Inverse agonist activity at human GAL4-fused RORalpha LBD transfected in 293T cell measured after 24 hrs by dual luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-alpha(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50005410(CHEMBL139197 | CHEMBL2137199)
Affinity DataIC50: 2.00E+4nMAssay Description:Inverse agonist activity at human GAL4-fused RORalpha LBD transfected in 293T cell measured after 24 hrs by dual luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetBile acid receptor(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610595(CHEMBL5279688)
Affinity DataIC50: 2.00E+4nMAssay Description:Inverse agonist activity at human GAL4-fused FXR LBD transfected in 293T cell measured after 24 hrs by dual luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetNuclear receptor ROR-alpha(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610599(CHEMBL5275972)
Affinity DataIC50: 2.00E+4nMAssay Description:Inverse agonist activity at human GAL4-fused RORalpha LBD transfected in 293T cell measured after 24 hrs by dual luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610597(CHEMBL5288443)
Affinity DataIC50: 2.00E+4nMAssay Description:Inverse agonist activity at human GAL4-fused LXRalpha LBD transfected in 293T cell measured after 24 hrs by dual luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetOxysterols receptor LXR-alpha(Human)
Guangzhou Medical University

Curated by ChEMBL
LigandPNGBDBM50610599(CHEMBL5275972)
Affinity DataIC50: 2.00E+4nMAssay Description:Inverse agonist activity at human GAL4-fused LXRalpha LBD transfected in 293T cell measured after 24 hrs by dual luciferase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
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