Compile Data Set for Download or QSAR
Report error Found 104 Enz. Inhib. hit(s) with all data for entry = 50013969
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571262(CHEMBL4858203)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571236(CHEMBL4871125)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571236(CHEMBL4871125)
Affinity DataIC50: 1.5nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571262(CHEMBL4858203)
Affinity DataIC50: 1.80nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571247(CHEMBL4866485)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571247(CHEMBL4866485)
Affinity DataIC50: 2.20nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571259(CHEMBL4849504)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571244(CHEMBL4846309)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571253(CHEMBL4867987)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571245(CHEMBL4875575)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571238(CHEMBL4856048)
Affinity DataKi:  2.90nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571244(CHEMBL4846309)
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571250(CHEMBL4847629)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571239(CHEMBL4874159)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571254(CHEMBL4867086)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571235(CHEMBL4872930)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50095293(CHEMBL3589085 | US9278953, 13)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571241(CHEMBL4867692)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571260(CHEMBL4854881)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571249(CHEMBL4867652)
Affinity DataKi:  5.70nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571237(CHEMBL4868434)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571245(CHEMBL4875575)
Affinity DataIC50: 5.90nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571250(CHEMBL4847629)
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571251(CHEMBL4849811)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571265(CHEMBL4857240)
Affinity DataKi:  7nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571261(CHEMBL4865327)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571263(CHEMBL4864985)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571260(CHEMBL4854881)
Affinity DataIC50: 8.10nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571259(CHEMBL4849504)
Affinity DataIC50: 8.70nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571255(CHEMBL4851344)
Affinity DataKi:  8.80nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571257(CHEMBL4874814)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571269(CHEMBL4865321)
Affinity DataKi:  9.40nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571238(CHEMBL4856048)
Affinity DataIC50: 9.70nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571271(CHEMBL4848523)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571269(CHEMBL4865321)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571242(CHEMBL4848264)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571266(CHEMBL4848372)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571253(CHEMBL4867987)
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571264(CHEMBL4872962)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571270(CHEMBL4873446)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571241(CHEMBL4867692)
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571252(CHEMBL4859300)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571254(CHEMBL4867086)
Affinity DataIC50: 14nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571246(CHEMBL4846915)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571256(CHEMBL4864757)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571274(CHEMBL4864589)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571237(CHEMBL4868434)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571268(CHEMBL4862628)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571271(CHEMBL4848523)
Affinity DataIC50: 17nMAssay Description:Antagonist activity at human EP3 receptor expressed in CHO cells by cell based cAMP functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50571279(CHEMBL4851298)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]PGE2 from human EP3 receptor expressed in CHO cells by radioligand competition binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
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