Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 50013621
TargetPeroxisome proliferator-activated receptor gamma(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568100(CHEMBL4861761)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARgamma expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568103(CHEMBL4847989)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARdelta expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568102(CHEMBL4847453)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARdelta expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568101(CHEMBL4870407)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARdelta expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568096(CHEMBL4866115)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARdelta expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568097(CHEMBL4879102)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARdelta expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568098(CHEMBL4877444)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARdelta expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568099(CHEMBL4855604)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARdelta expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor delta(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568100(CHEMBL4861761)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARdelta expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568103(CHEMBL4847989)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARgamma expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568102(CHEMBL4847453)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARgamma expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568101(CHEMBL4870407)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARgamma expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568096(CHEMBL4866115)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARgamma expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568097(CHEMBL4879102)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARgamma expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568098(CHEMBL4877444)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARgamma expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568099(CHEMBL4855604)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at Gal4-fused human PPARgamma expressed in monkey CV1 cells assessed as receptor transactivation incubated for 45 hrs by luciferase ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568096(CHEMBL4866115)
Affinity DataEC50:  0.850nMAssay Description:Agonist activity at Gal4-fused human PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568103(CHEMBL4847989)
Affinity DataEC50:  20nMAssay Description:Agonist activity at Gal4-fused mouse PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568102(CHEMBL4847453)
Affinity DataEC50:  10nMAssay Description:Agonist activity at Gal4-fused mouse PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568101(CHEMBL4870407)
Affinity DataEC50:  30nMAssay Description:Agonist activity at Gal4-fused mouse PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568096(CHEMBL4866115)
Affinity DataEC50:  3nMAssay Description:Agonist activity at Gal4-fused mouse PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568097(CHEMBL4879102)
Affinity DataEC50:  10nMAssay Description:Agonist activity at Gal4-fused mouse PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568098(CHEMBL4877444)
Affinity DataEC50:  20nMAssay Description:Agonist activity at Gal4-fused mouse PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568099(CHEMBL4855604)
Affinity DataEC50:  20nMAssay Description:Agonist activity at Gal4-fused mouse PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Mouse)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568100(CHEMBL4861761)
Affinity DataEC50:  3nMAssay Description:Agonist activity at Gal4-fused mouse PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568103(CHEMBL4847989)
Affinity DataEC50:  12nMAssay Description:Agonist activity at Gal4-fused human PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568102(CHEMBL4847453)
Affinity DataEC50:  1nMAssay Description:Agonist activity at Gal4-fused human PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568101(CHEMBL4870407)
Affinity DataEC50:  3nMAssay Description:Agonist activity at Gal4-fused human PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568100(CHEMBL4861761)
Affinity DataEC50:  0.870nMAssay Description:Agonist activity at Gal4-fused human PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568099(CHEMBL4855604)
Affinity DataEC50:  1nMAssay Description:Agonist activity at Gal4-fused human PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568098(CHEMBL4877444)
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at Gal4-fused human PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
City of Hope National Medical Center

Curated by ChEMBL
LigandPNGBDBM50568097(CHEMBL4879102)
Affinity DataEC50:  0.950nMAssay Description:Agonist activity at Gal4-fused human PPARalpha co-expressed with RXRalpha in monkey CV1 cells assessed as PPRE transcriptional activation incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed