Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50016595
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595940(CHEMBL5197924)
Affinity DataEC50: >1.00E+5nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595948(CHEMBL5205628)
Affinity DataEC50:  790nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595947(CHEMBL5182239)
Affinity DataEC50:  1.20E+3nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595946(CHEMBL5180168)
Affinity DataEC50:  3.60E+3nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595945(CHEMBL5178739)
Affinity DataEC50:  1.70E+3nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595939(CHEMBL5209370)
Affinity DataEC50:  1.80E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595938(CHEMBL5197292)
Affinity DataEC50:  3.10E+3nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595944(CHEMBL5177875)
Affinity DataEC50:  5.80E+3nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50519883(CHEMBL4522217)
Affinity DataEC50:  8.20E+3nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595943(CHEMBL5189438)
Affinity DataEC50:  1.50E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595942(CHEMBL5177120)
Affinity DataEC50:  7.50E+3nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595941(CHEMBL5200206)
Affinity DataEC50:  2.50E+3nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50106301(CHEMBL3598140)
Affinity DataEC50:  340nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment by T...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50106301(CHEMBL3598140)
Affinity DataIC50: 7nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595941(CHEMBL5200206)
Affinity DataIC50: 7.40nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595938(CHEMBL5197292)
Affinity DataIC50: 12nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50106301(CHEMBL3598140)
Affinity DataIC50: 13nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595941(CHEMBL5200206)
Affinity DataIC50: 20nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595938(CHEMBL5197292)
Affinity DataIC50: 31nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595946(CHEMBL5180168)
Affinity DataIC50: 33nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595945(CHEMBL5178739)
Affinity DataIC50: 46nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595944(CHEMBL5177875)
Affinity DataIC50: 74nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50519883(CHEMBL4522217)
Affinity DataIC50: 100nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595946(CHEMBL5180168)
Affinity DataIC50: 110nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595945(CHEMBL5178739)
Affinity DataIC50: 140nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595944(CHEMBL5177875)
Affinity DataIC50: 220nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50519883(CHEMBL4522217)
Affinity DataIC50: 270nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595942(CHEMBL5177120)
Affinity DataIC50: 290nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595942(CHEMBL5177120)
Affinity DataIC50: 490nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595943(CHEMBL5189438)
Affinity DataIC50: 1.50E+3nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595948(CHEMBL5205628)
Affinity DataIC50: 1.80E+3nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595947(CHEMBL5182239)
Affinity DataIC50: 1.90E+3nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595939(CHEMBL5209370)
Affinity DataIC50: 2.50E+3nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595948(CHEMBL5205628)
Affinity DataIC50: 2.90E+3nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595947(CHEMBL5182239)
Affinity DataIC50: 3.30E+3nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595943(CHEMBL5189438)
Affinity DataIC50: 3.60E+3nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595940(CHEMBL5197924)
Affinity DataIC50: 6.20E+3nMAssay Description:Displacement of Alexa flour647-labeled MRL-871 from RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) cell...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50106301(CHEMBL3598140)
Affinity DataIC50: 6.30E+3nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetNuclear receptor ROR-gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595939(CHEMBL5209370)
Affinity DataIC50: 6.60E+3nMAssay Description:Allosteric inverse agonist activity at C-terminal His-tagged RORgammat LBD (265 to 507 residues) (unknown origin) expressed in Escherichia coli BL21(...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595948(CHEMBL5205628)
Affinity DataIC50: 1.90E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595947(CHEMBL5182239)
Affinity DataIC50: 2.00E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595945(CHEMBL5178739)
Affinity DataIC50: 2.90E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595938(CHEMBL5197292)
Affinity DataIC50: 6.30E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595941(CHEMBL5200206)
Affinity DataIC50: 6.40E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595944(CHEMBL5177875)
Affinity DataIC50: 6.70E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595946(CHEMBL5180168)
Affinity DataIC50: 7.90E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50519883(CHEMBL4522217)
Affinity DataIC50: 8.10E+4nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595943(CHEMBL5189438)
Affinity DataIC50: 1.00E+5nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595942(CHEMBL5177120)
Affinity DataIC50: 1.00E+5nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
Technische Universiteit Eindhoven

Curated by ChEMBL
LigandPNGBDBM50595940(CHEMBL5197924)
Affinity DataIC50: 1.00E+5nMAssay Description:Inverse agonist activity at His6-tagged PPARgamma LBD (unknown origin) assessed as N-terminal biotinylated PGC1a coactivator peptide recruitment in p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
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