Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50014447
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50576337(CHEMBL4877326)
Affinity DataIC50: 790nMAssay Description:Displacement of Alexafluor 647-conjugated PFI-1 from N-terminal-His6-tagged human BRD4 BD1 domain (44 to 170 residues) incubated for 30 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50576336(CHEMBL4849738)
Affinity DataIC50: 2.42E+3nMAssay Description:Displacement of Alexafluor 647-conjugated PFI-1 from N-terminal-His6-tagged human BRD4 BD1 domain (44 to 170 residues) incubated for 30 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50576335(CHEMBL4864626)
Affinity DataIC50: 1.18E+4nMAssay Description:Displacement of Alexafluor 647-conjugated PFI-1 from N-terminal-His6-tagged human BRD4 BD1 domain (44 to 170 residues) incubated for 30 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50576334(CHEMBL4845767)
Affinity DataIC50: 3.00E+4nMAssay Description:Displacement of Alexafluor 647-conjugated PFI-1 from N-terminal-His6-tagged human BRD4 BD1 domain (44 to 170 residues) incubated for 30 mins by fluor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed