Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50013941
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50571076(CHEMBL4860842)
Affinity DataKd:  480nMAssay Description:Inhibition of human wild type RIPK1 (M1 to K305) expressed in bacterial system by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50571077(CHEMBL4869920)
Affinity DataKd:  1.70E+3nMAssay Description:Inhibition of human wild type RIPK1 (M1 to K305) expressed in bacterial system by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50571078(CHEMBL4850219)
Affinity DataKd:  430nMAssay Description:Inhibition of human wild type RIPK1 (M1 to K305) expressed in bacterial system by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM99471(US8497274, 32)
Affinity DataKd:  480nMAssay Description:Inhibition of human wild type RIPK1 (M1 to K305) expressed in bacterial system by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50528231(CHEMBL4540715)
Affinity DataKd:  97nMAssay Description:Inhibition of human wild type RIPK1 (M1 to K305) expressed in bacterial system by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50571076(CHEMBL4860842)
Affinity DataKd:  270nMAssay Description:Inhibition of human wild type RIPK3 (M1 to Q307) expressed in bacterial system by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50571077(CHEMBL4869920)
Affinity DataKd:  650nMAssay Description:Inhibition of human wild type RIPK3 (M1 to Q307) expressed in bacterial system by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50571078(CHEMBL4850219)
Affinity DataKd:  145nMAssay Description:Inhibition of human wild type RIPK3 (M1 to Q307) expressed in bacterial system by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM99471(US8497274, 32)
Affinity DataKd:  105nMAssay Description:Inhibition of human wild type RIPK3 (M1 to Q307) expressed in bacterial system by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 3(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50528231(CHEMBL4540715)
Affinity DataKd:  77nMAssay Description:Inhibition of human wild type RIPK3 (M1 to Q307) expressed in bacterial system by kinomescan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50513004(CHEMBL4521353)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of GST-tagged RIPK1 (1 to 375) (unknown origin) incubated for 4 hrs by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50513004(CHEMBL4521353)
Affinity DataIC50: 16nMAssay Description:Inhibition of GST-tagged RIPK1 (1 to 375) (unknown origin) by fluorescent polarization based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50513014(CHEMBL4442060)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-tagged RIPK1 (1 to 375) (unknown origin) by fluorescent polarization based binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Ningxia Medical University

Curated by ChEMBL
LigandPNGBDBM50513014(CHEMBL4442060)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of GST-tagged RIPK1 (1 to 375) (unknown origin) incubated for 4 hrs by ADP-Glo kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed