Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 50014993
TargetDual specificity protein kinase TTK(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50581714(CHEMBL5092617)
Affinity DataIC50: 3.20nMAssay Description:Inhibition of human hexa-His tagged MPS1 (515 to 795 residue) expressed in Escherichia coli BL2I-DE3 cells incubated for 4 hrs in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetDual specificity protein kinase TTK(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50581717(CHEMBL5093783)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human hexa-His tagged MPS1 (515 to 795 residue) expressed in Escherichia coli BL2I-DE3 cells incubated for 4 hrs in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetDual specificity protein kinase TTK(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50581716(CHEMBL5080463)
Affinity DataIC50: 6.30nMAssay Description:Inhibition of human hexa-His tagged MPS1 (515 to 795 residue) expressed in Escherichia coli BL2I-DE3 cells incubated for 4 hrs in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetDual specificity protein kinase TTK(Human)
Yonsei University

Curated by ChEMBL
LigandPNGBDBM50581715(CHEMBL5092060)
Affinity DataIC50: 6.40nMAssay Description:Inhibition of human hexa-His tagged MPS1 (515 to 795 residue) expressed in Escherichia coli BL2I-DE3 cells incubated for 4 hrs in presence of ATP by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMedPDB3D3D Structure (crystal)