Report error Found 97 Enz. Inhib. hit(s) with all data for entry = 50013996
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 832nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 6.61E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 1.38E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 1.18E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 933nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 1.59E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 1.74E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 468nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 98nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 25nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 39nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 1.62E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 7.59E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 468nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 5.13E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 158nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 447nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 158nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 102nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 4(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 3.16E+3nMAssay Description:Agonist activity at human TRPM4 expressed in CHO cells assessed as increase in A23187-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 4(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <6.31E+4nMAssay Description:Agonist activity at human TRPM4 expressed in CHO cells assessed as increase in A23187-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 4(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <6.31E+4nMAssay Description:Agonist activity at human TRPM4 expressed in CHO cells assessed as increase in A23187-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 4(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <6.31E+4nMAssay Description:Agonist activity at human TRPM4 expressed in CHO cells assessed as increase in A23187-induced intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Mouse)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Agonist activity at mouse TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Mouse)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 44nMAssay Description:Agonist activity at mouse TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Mouse)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 85nMAssay Description:Agonist activity at mouse TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Mouse)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 891nMAssay Description:Agonist activity at mouse TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 6.03E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by QPatch HTX assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 309nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 295nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 85nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 38nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 29nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 18nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 7.90nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 1.45E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <3.16E+4nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 44nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 5.25E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 5(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: 2.82E+3nMAssay Description:Agonist activity at human TRPM5 expressed in CHO-K1 cells maintained at 80 mV final holding potential by syncroPatch assayMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily M member 8(Human)
Aptuit, An Evotec
Curated by ChEMBL
Aptuit, An Evotec
Curated by ChEMBL
Affinity DataEC50: <1.58E+4nMAssay Description:Agonist activity at human TRPM8 expressed in HEK cells assessed as increase in menthol-induced intracellular calcium level measured after 1 hr by FLI...More data for this Ligand-Target Pair










































