Compile Data Set for Download or QSAR
Report error Found 83 Enz. Inhib. hit(s) with all data for entry = 50013995
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataKd:  21nMAssay Description:Binding affinity to human CBP measured at 15 degreeC by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataKd:  850nMAssay Description:Binding affinity to human BRD4 measured at 15 degreeC by ITC assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571557(CHEMBL4853072)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human partial length BRD4 bromodomain 1 long isoform (N44 to E168 residues) expressed in bacterial expression system by BromoELEC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571550(CHEMBL4867046)
Affinity DataKd:  9.20E+3nMAssay Description:Binding affinity to human partial length BRD4 bromodomain 1 long isoform (N44 to E168 residues) expressed in bacterial expression system by BromoELEC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571569(CHEMBL4875989)
Affinity DataKd:  1.30E+4nMAssay Description:Binding affinity to human partial length EP300 (A1040 to G1161 residues) expressed in bacterial expression system by BromoELECT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571557(CHEMBL4853072)
Affinity DataKd:  215nMAssay Description:Binding affinity to human partial length EP300 (A1040 to G1161 residues) expressed in bacterial expression system by BromoELECT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetHistone acetyltransferase p300(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571550(CHEMBL4867046)
Affinity DataKd:  285nMAssay Description:Binding affinity to human partial length EP300 (A1040 to G1161 residues) expressed in bacterial expression system by BromoELECT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571557(CHEMBL4853072)
Affinity DataKd:  315nMAssay Description:Binding affinity to human partial length CREBBP (R1081 to G1197 residues) expressed in bacterial expression system by BromoELECT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571550(CHEMBL4867046)
Affinity DataKd:  265nMAssay Description:Binding affinity to human partial length CREBBP (R1081 to G1197 residues) expressed in bacterial expression system by BromoELECT assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataIC50: 28nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataIC50: 64nMAssay Description:Inhibition of human CBP by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571557(CHEMBL4853072)
Affinity DataIC50: 72nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM188517(PF-CBP1)
Affinity DataIC50: 130nMAssay Description:Inhibition of CBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571550(CHEMBL4867046)
Affinity DataIC50: 159nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571553(CHEMBL4859434)
Affinity DataIC50: 214nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571551(CHEMBL4875068)
Affinity DataIC50: 290nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50151661(CHEMBL3752296)
Affinity DataIC50: 323nMAssay Description:Inhibition of CBP (unknown origin) by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571549(CHEMBL4878741)
Affinity DataIC50: 460nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571542(CHEMBL4878894)
Affinity DataIC50: 507nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571544(CHEMBL4877061)
Affinity DataIC50: 510nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571554(CHEMBL4875619)
Affinity DataIC50: 633nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571541(CHEMBL4848215)
Affinity DataIC50: 718nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571566(CHEMBL4876541)
Affinity DataIC50: 750nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571548(CHEMBL4864701)
Affinity DataIC50: 923nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571547(CHEMBL4848135)
Affinity DataIC50: 950nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571538(CHEMBL4868314)
Affinity DataIC50: 1.17E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571556(CHEMBL4863302)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571546(CHEMBL4864355)
Affinity DataIC50: 1.88E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571555(CHEMBL4861811)
Affinity DataIC50: 1.92E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571536(CHEMBL4846628)
Affinity DataIC50: 2.21E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571552(CHEMBL4865121)
Affinity DataIC50: 2.33E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571563(CHEMBL4866716)
Affinity DataIC50: 2.53E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571546(CHEMBL4864355)
Affinity DataIC50: 2.77E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571538(CHEMBL4868314)
Affinity DataIC50: 2.95E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571545(CHEMBL4861666)
Affinity DataIC50: 3.02E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571542(CHEMBL4878894)
Affinity DataIC50: 3.38E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571549(CHEMBL4878741)
Affinity DataIC50: 3.42E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571567(CHEMBL4847433)
Affinity DataIC50: 3.51E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571559(CHEMBL4867415)
Affinity DataIC50: 4.95E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571557(CHEMBL4853072)
Affinity DataIC50: 5.19E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571547(CHEMBL4848135)
Affinity DataIC50: 5.63E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571558(CHEMBL4864902)
Affinity DataIC50: 6.07E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571566(CHEMBL4876541)
Affinity DataIC50: 6.21E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571553(CHEMBL4859434)
Affinity DataIC50: 6.48E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571550(CHEMBL4867046)
Affinity DataIC50: 6.59E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571548(CHEMBL4864701)
Affinity DataIC50: 7.11E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571541(CHEMBL4848215)
Affinity DataIC50: 7.43E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571543(CHEMBL4855910)
Affinity DataIC50: 7.55E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM50571540(CHEMBL4854416)
Affinity DataIC50: 7.83E+3nMAssay Description:Inhibition of His-tagged CBP (unknown origin) using biotinylated-H3K56ac peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
University of Massachusetts Boston

Curated by ChEMBL
LigandPNGBDBM188519(SGC-CBP30)
Affinity DataIC50: 7.94E+3nMAssay Description:Inhibition of His-tagged BRD4 BD1 (unknown origin) using biotinylated-JQ1 peptide as substrate incubated for 1 hr by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
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