Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50013785
TargetCytochrome P450 3A4(Human)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50569646(Azamulin)
Affinity DataIC50: 240nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using testosterone as substrate incubated for 10 mins by LC/MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50569645(CHEBI:44137 | Tiamulin | SO 14055 | SQ 14055 | SQ-...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using testosterone as substrate incubated for 5 mins followed by NADPH addition and measured after 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetCytochrome P450 3A4(Human)
South China Agricultural University

Curated by ChEMBL
LigandPNGBDBM50569644(CHEMBL4856492)
Affinity DataIC50: 3.95E+3nMAssay Description:Inhibition of CYP3A4 in human liver microsomes using testosterone as substrate incubated for 5 mins followed by NADPH addition and measured after 5 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed