Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50018242
TargetFree fatty acid receptor 1(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM22496(CHEMBL207881 | 3-(4-{[(3-phenoxyphenyl)methyl]amin...)
Affinity DataEC50:  48nMAssay Description:Agonist activity at GPR40 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetFree fatty acid receptor 4(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM22496(CHEMBL207881 | 3-(4-{[(3-phenoxyphenyl)methyl]amin...)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at GPR120 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetFree fatty acid receptor 4(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50408137(CHEMBL5275980)
Affinity DataEC50:  165nMAssay Description:Agonist activity at human GPR120 expressed in HEK293 cells assessed as calcium accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetFree fatty acid receptor 4(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50408137(CHEMBL5275980)
Affinity DataEC50:  125nMAssay Description:Agonist activity at human GPR120 expressed in HEK293 cells by beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetFree fatty acid receptor 4(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50408138(CHEMBL5286838)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as calcium accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetFree fatty acid receptor 4(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50408138(CHEMBL5286838)
Affinity DataEC50:  5.30nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells by beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetFree fatty acid receptor 4(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50408138(CHEMBL5286838)
Affinity DataEC50:  60nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetFree fatty acid receptor 4(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM382129(4-(4-((4'-cyclopropyl-3,4,5,6-tetrahydro-[1,1'-bip...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetFree fatty acid receptor 4(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM382131(4-(4-((2-(5,6,7,8-tetrahydronaphthalen-2-yl)cycloh...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetFree fatty acid receptor 4(Human)
University of Siena

Curated by ChEMBL
LigandPNGBDBM50408139(CHEMBL5272316)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human GPR120 expressed in CHO-K1 cells by BRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed