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Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50015612
TargetSerine/threonine-protein kinase PLK1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50435727(CHEMBL2392545)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMedPDB3D3D Structure (crystal)
TargetSerine/threonine-protein kinase PLK1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM25121(4-{[(7R)-8-cyclopentyl-7-ethyl-5-methyl-6-oxo-5,6,...)
Affinity DataIC50: 0.830nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human PLK1 (1 to 603 residues) expressed in baculovirus expression system incubated for 45 mins using...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50587787(CHEMBL5190855)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of PLK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50587788(CHEMBL5175599)
Affinity DataIC50: 267nMAssay Description:Inhibition of PLK1-PBD (unknown origin) using FITC-GPMQSpTPLNG-OH as substrate measured after 30 mins by Fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50403017(CHEMBL2207846)
Affinity DataKd:  445nMAssay Description:Binding affinity to recombinant N-terminal His6-DsRed tagged PLK1-PBD (unknown origin) expressed in Escherichia coli BL21(DE3) Rosetta cells by ITC a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50587789(CHEMBL5188203)
Affinity DataKd:  1.28E+4nMAssay Description:Binding affinity to human PLK1-PBD (326 to 603 residues) expressed in Escherichia coli BL21(DE3) rosetta cells by microscale thermophoresis analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50587789(CHEMBL5188203)
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of human PLK1-PBD (326 to 603 residues) expressed in Escherichia coli BL21(DE3) rosetta cells using 5-carboxyfluorescein-GPMQSpTPLNG-OH as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50587786(CHEMBL5192049)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of human PLK1-PBD expressed in Escherichia coli BL21(DE3) rosetta cells using 5-carboxyfluorescein-GPMQSpTPLNG-OH as substrate preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50587786(CHEMBL5192049)
Affinity DataIC50: 1.79E+4nMAssay Description:Inhibition of human PLK1-PBD expressed in Escherichia coli BL21(DE3) rosetta cells using 5-carboxyfluorescein-GPMQSpTPLNG-OH as substrate preincubate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK2(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50587786(CHEMBL5192049)
Affinity DataIC50: 9.55E+7nMAssay Description:Inhibition of recombinant C-terminal 6His-tagged human PLK2-PBD expressed in Escherichia coli BL21(DE3) rosetta cells using 5-carboxyfluorescein-GPMQ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase PLK3(Human)
Shandong First Medical University & Shandong Academy of Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50587786(CHEMBL5192049)
Affinity DataIC50: 1.00E+8nMAssay Description:Inhibition of recombinant N-terminal MBP-tagged human PLK3-PBD expressed in Escherichia coli BL21(DE3) rosetta cells using 5-carboxyfluorescein-GPLAT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/18/2023
Entry Details
PubMed