Compile Data Set for Download or QSAR
Report error Found 33 Enz. Inhib. hit(s) with all data for entry = 50013209
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563723(CHEMBL4128865)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of wild-type human CK1delta using PLSRTLpSVASLPGL as substrate incubated for 40 mins in presence of ATP by Kinase-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform epsilon(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50364141(CHEMBL1951415)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of full-length human CK1epsilon expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells using PLSRTLpSVASLPGL as substrate i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50364141(CHEMBL1951415)
Affinity DataIC50: 14nMAssay Description:Inhibition of full-length human CK1delta expressed in Escherichia coli BL21-CodonPlus(DE3)-RIL competent cells using PLSRTLpSVASLPGL as substrate inc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform epsilon(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563723(CHEMBL4128865)
Affinity DataIC50: 17nMAssay Description:Inhibition of wild-type human CK1epsilon using PLSRTLpSVASLPGL as substrate incubated for 70 mins in presence of ATP by Kinase-Glo luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563717(CHEMBL4742954)
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563710(CHEMBL4793727)
Affinity DataIC50: 210nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563711(CHEMBL4793501)
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563717(CHEMBL4742954)
Affinity DataIC50: 300nMAssay Description:Inhibition of recombinant human full-length N-terminal GST-tagged CK1delta using casein as substrate measured after 10 mins in presence of ATP by Kin...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563706(CHEMBL4776464)
Affinity DataIC50: 320nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563714(CHEMBL4760165)
Affinity DataIC50: 460nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563719(CHEMBL4784755)
Affinity DataIC50: 470nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563704(CHEMBL4752690)
Affinity DataIC50: 480nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563720(CHEMBL4745216)
Affinity DataIC50: 530nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563721(CHEMBL4782184)
Affinity DataIC50: 670nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563712(CHEMBL4795601)
Affinity DataIC50: 740nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563718(CHEMBL4793180)
Affinity DataIC50: 750nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563716(CHEMBL4783829)
Affinity DataIC50: 910nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563707(CHEMBL4761245)
Affinity DataIC50: 990nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563709(CHEMBL4744604)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563713(CHEMBL4783769)
Affinity DataIC50: 1.32E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563702(CHEMBL4785118)
Affinity DataIC50: 2.06E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563722(CHEMBL4743699)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563703(CHEMBL4752279)
Affinity DataIC50: 4.75E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563708(CHEMBL4743742)
Affinity DataIC50: 5.32E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563715(CHEMBL4758938)
Affinity DataIC50: 5.65E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563697(CHEMBL4754212)
Affinity DataIC50: 8.67E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563696(CHEMBL4747427)
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563695(CHEMBL4790041)
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563700(CHEMBL4800506)
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563701(CHEMBL4762847)
Affinity DataIC50: 1.66E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563698(CHEMBL4758812)
Affinity DataIC50: 2.02E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563699(CHEMBL4747963)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetCasein kinase I isoform delta(Human)
University of Trieste

Curated by ChEMBL
LigandPNGBDBM50563705(CHEMBL4789473)
Affinity DataIC50: 2.68E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged CK1delta (1 to 294 residues) using casein as substrate measured after 60 mins in presence of AT...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed