Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50013192
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563455(CHEMBL4751616)
Affinity DataEC50:  107nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50244791((2-Fluoro-4-methanesulfonyl-phenyl)-{6-[4-(3-isopr...)
Affinity DataEC50:  6nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563462(CHEMBL4789532)
Affinity DataEC50:  153nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563461(CHEMBL4743968)
Affinity DataEC50:  106nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563460(CHEMBL4790469)
Affinity DataEC50:  720nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563459(CHEMBL4790521)
Affinity DataEC50:  125nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563458(CHEMBL4784457)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563457(CHEMBL4796294)
Affinity DataEC50:  819nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563456(CHEMBL4778466)
Affinity DataEC50:  1.87E+3nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563447(CHEMBL4782568)
Affinity DataEC50:  1.41E+3nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563454(CHEMBL4760659)
Affinity DataEC50:  805nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563453(CHEMBL4777445)
Affinity DataEC50:  745nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563452(CHEMBL4748865)
Affinity DataEC50:  75nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563451(CHEMBL4779985)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563450(CHEMBL4741006)
Affinity DataEC50:  88nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563449(CHEMBL4755177)
Affinity DataEC50:  790nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetGlucose-dependent insulinotropic receptor(Human)
M. S. University of Baroda

Curated by ChEMBL
LigandPNGBDBM50563448(CHEMBL4744049)
Affinity DataEC50:  157nMAssay Description:Agonist activity at human GPR119 stably transfected in CHO-K1 cells assessed as increase in cAMP stimulation after 1 hr by enzyme immunoassayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed