Compile Data Set for Download or QSAR
Report error Found 140 Enz. Inhib. hit(s) with all data for entry = 50013859
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the later state of compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570357(CHEMBL4865147)
Affinity DataIC50: 55nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the later state of compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50: 60nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in HEK293 cells assessed as reduction in glycine-induced currents by whol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570358(CHEMBL4855686)
Affinity DataIC50: 67nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the later state of compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570341(CHEMBL4849489)
Affinity DataIC50: 90nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570346(CHEMBL4870499)
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570342(CHEMBL4857611)
Affinity DataIC50: 130nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50: 134nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the onset of compound app...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570355(CHEMBL4873527)
Affinity DataIC50: 137nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the later state of compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50: 150nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50: 151nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570356(CHEMBL4864603)
Affinity DataIC50: 158nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the later state of compou...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570343(CHEMBL4851242)
Affinity DataIC50: 170nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570340(CHEMBL4865584)
Affinity DataIC50: 204nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570340(CHEMBL4865584)
Affinity DataIC50: 210nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570344(CHEMBL4848356)
Affinity DataIC50: 400nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570340(CHEMBL4865584)
Affinity DataIC50: 427nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570340(CHEMBL4865584)
Affinity DataIC50: 430nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50: 510nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570341(CHEMBL4849489)
Affinity DataIC50: 510nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)
Affinity DataIC50: 513nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570341(CHEMBL4849489)
Affinity DataIC50: 513nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570333(CHEMBL4870655)
Affinity DataIC50: 676nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570333(CHEMBL4870655)
Affinity DataIC50: 680nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570339(CHEMBL4850957)
Affinity DataIC50: 720nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570345(CHEMBL4870669)
Affinity DataIC50: 730nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570345(CHEMBL4870669)
Affinity DataIC50: 741nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570341(CHEMBL4849489)
Affinity DataIC50: 776nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570341(CHEMBL4849489)
Affinity DataIC50: 780nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570339(CHEMBL4850957)
Affinity DataIC50: 800nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in HEK293 cells assessed as reduction in glycine-induced currents by whol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570355(CHEMBL4873527)
Affinity DataIC50: 852nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the onset of compound app...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570345(CHEMBL4870669)
Affinity DataIC50: 871nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570345(CHEMBL4870669)
Affinity DataIC50: 880nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570339(CHEMBL4850957)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570339(CHEMBL4850957)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570337(CHEMBL4860026)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570333(CHEMBL4870655)
Affinity DataIC50: 1.20E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570333(CHEMBL4870655)
Affinity DataIC50: 1.23E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570337(CHEMBL4860026)
Affinity DataIC50: 1.30E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in HEK293 cells assessed as reduction in glycine-induced currents by whol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570357(CHEMBL4865147)
Affinity DataIC50: 1.34E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the onset of compound app...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570351(CHEMBL4873219)
Affinity DataIC50: 1.40E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570338(CHEMBL4849060)
Affinity DataIC50: 1.50E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570347(CHEMBL4864670)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570347(CHEMBL4864670)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in human tsA201 cells assessed as reduction in glycine-induced response incub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570344(CHEMBL4848356)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570350(CHEMBL4849579)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570344(CHEMBL4848356)
Affinity DataIC50: 1.74E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570339(CHEMBL4850957)
Affinity DataIC50: 1.78E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
TargetGlycine receptor subunit alpha-1/beta(Human)
The German University In Cairo

Curated by ChEMBL
LigandPNGBDBM50570357(CHEMBL4865147)
Affinity DataIC50: 1.78E+3nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in human tsA201 cells assessed as reduction in glycine-induced response i...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/20/2022
Entry Details Article
PubMed
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