Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 50012405
TargetP2X purinoceptor 7(Human)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50557382(CHEMBL4780724)
Affinity DataIC50: 6.00E+3nMAssay Description:Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as reduction in benzoyl-ATP-induced YO-PRO-1 dye uptake pre-incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50557380(CHEMBL4751055)
Affinity DataIC50: 9.00E+3nMAssay Description:Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as reduction in benzoyl-ATP-induced YO-PRO-1 dye uptake pre-incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50557381(CHEMBL4757539)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as reduction in benzoyl-ATP-induced YO-PRO-1 dye uptake pre-incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50557385(CHEMBL4780725)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as reduction in benzoyl-ATP-induced YO-PRO-1 dye uptake pre-incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50557384(CHEMBL4743642)
Affinity DataIC50: 1.02E+4nMAssay Description:Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as reduction in benzoyl-ATP-induced YO-PRO-1 dye uptake pre-incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50557383(CHEMBL4753833)
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as reduction in benzoyl-ATP-induced YO-PRO-1 dye uptake pre-incubated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetP2X purinoceptor 7(Human)
Universidad Aut£Noma De Madrid

Curated by ChEMBL
LigandPNGBDBM50557380(CHEMBL4751055)
Affinity DataIC50: 1.37E+4nMAssay Description:Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as reduction in benzoyl-ATP-induced intracellular Ca2+ level by Fura-2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed