Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50013140
LigandPNGBDBM50193709(CHEMBL3911017)
Affinity DataIC50: 17nMAssay Description:Inhibition of wild type EZH2 in human KARPAS-422 cells assessed as effect on H3K27Me3 levelsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
LigandPNGBDBM50562994(CHEMBL4740532)
Affinity DataIC50: 30nMAssay Description:Inhibition of wild type EZH2 in human KARPAS-422 cells assessed as effect on H3K27Me3 levelsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
LigandPNGBDBM50193709(CHEMBL3911017)
Affinity DataKi:  1nMAssay Description:Inhibition of wild type EZH2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
LigandPNGBDBM50562994(CHEMBL4740532)
Affinity DataKi:  2nMAssay Description:Inhibition of wild type EZH2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
LigandPNGBDBM50193709(CHEMBL3911017)
Affinity DataKi:  3nMAssay Description:Inhibition of wild type EZH2 Y641N mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
LigandPNGBDBM50562994(CHEMBL4740532)
Affinity DataKi:  7nMAssay Description:Inhibition of wild type EZH2 Y641N mutant (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed