Compile Data Set for Download or QSAR
Report error Found 70 Enz. Inhib. hit(s) with all data for entry = 50012007
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553217(CHEMBL4761747)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553212(CHEMBL4763380)
Affinity DataIC50: 10nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 18nMAssay Description:Inhibition of human NEK2 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553200(CHEMBL4796125)
Affinity DataIC50: 26nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553205(CHEMBL4743876)
Affinity DataIC50: 39nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553213(CHEMBL4779487)
Affinity DataIC50: 42nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553201(CHEMBL4775990)
Affinity DataIC50: 50nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553215(CHEMBL4783060)
Affinity DataIC50: 57nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553198(CHEMBL4796754)
Affinity DataIC50: 57nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 62nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553204(CHEMBL4748191)
Affinity DataIC50: 64nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553199(CHEMBL4795738)
Affinity DataIC50: 71nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553197(CHEMBL4746054)
Affinity DataIC50: 72nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553196(CHEMBL4783265)
Affinity DataIC50: 76nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553214(CHEMBL4776787)
Affinity DataIC50: 76nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553195(CHEMBL4746829)
Affinity DataIC50: 79nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 80nMAssay Description:Inhibition of Aurora A (unknown origin) preincubated with enzyme for 15 mins followed by substrate/ATP challenge for 90 mins by ProfilerPro plate bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553209(CHEMBL4761123)
Affinity DataIC50: 88nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553208(CHEMBL4776060)
Affinity DataIC50: 93nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553210(CHEMBL4754015)
Affinity DataIC50: 100nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553203(CHEMBL4756141)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553202(CHEMBL4753609)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553194(CHEMBL4759854)
Affinity DataIC50: 116nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNUAK family SNF1-like kinase 1(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 120nMAssay Description:Inhibition of human NAUK1 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553216(CHEMBL4754958)
Affinity DataIC50: 130nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235361(CHEMBL4074015)
Affinity DataIC50: 140nMAssay Description:Inhibition of human NEK2 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235361(CHEMBL4074015)
Affinity DataIC50: 140nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235350(CHEMBL4094562)
Affinity DataIC50: 140nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235350(CHEMBL4094562)
Affinity DataIC50: 150nMAssay Description:Inhibition of human NEK2 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553206(CHEMBL4751371)
Affinity DataIC50: 210nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 220nMAssay Description:Inhibition of human JAK2 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 7(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 240nMAssay Description:Inhibition of human TAK1 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 9(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 270nMAssay Description:Inhibition of human MLK1 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase kinase kinase 11(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 320nMAssay Description:Inhibition of human MLK3 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDual specificity mitogen-activated protein kinase kinase 1(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 550nMAssay Description:Inhibition of human MKK1 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 560nMAssay Description:Inhibition of human ChK1 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase TBK1(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 740nMAssay Description:Inhibition of human TBK1 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50347863(CHEMBL1802870)
Affinity DataIC50: 770nMAssay Description:Inhibition of NEK2 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553211(CHEMBL4785527)
Affinity DataIC50: 820nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCytoplasmic tyrosine-protein kinase BMX(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553207(CHEMBL4786783)
Affinity DataIC50: 830nMAssay Description:Inhibition of BMX (unknown origin) preincubated with enzyme for 15 mins followed by substrate/ATP challenge for 90 mins by ProfilerPro plate based la...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235350(CHEMBL4094562)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human Aurora A by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235361(CHEMBL4074015)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of human ChK2 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase beta-1(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235361(CHEMBL4074015)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of human P70S6K by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235350(CHEMBL4094562)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of human ChK2 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235361(CHEMBL4074015)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human ChK1 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetGlycogen synthase kinase-3 beta(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235350(CHEMBL4094562)
Affinity DataIC50: 7.40E+3nMAssay Description:Inhibition of human GSK-3beta by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235361(CHEMBL4074015)
Affinity DataIC50: 9.60E+3nMAssay Description:Inhibition of human CDK1 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProto-oncogene tyrosine-protein kinase Src(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235350(CHEMBL4094562)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of human SRC by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Chk1(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50235350(CHEMBL4094562)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human ChK1 by kinase-profiling analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase Nek2(Human)
Newcastle University

Curated by ChEMBL
LigandPNGBDBM50553218(CHEMBL4755796)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of human recombinant full length His-tagged NEK2 expressed in baculovirus expression system assessed as inhibition of substrate phosphoryl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
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