Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 50012002
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50008099(CHEMBL1234777)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50008099(CHEMBL1234777)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of recombinant human liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50350311(CHEMBL1812661)
Affinity DataIC50: 1.68E+4nMAssay Description:Inhibition of recombinant human ARG1 expressed in CHO-K1 cells assessed as reduction in urea level incubated for 24 hrs by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50045936(CHEMBL69863 | 4-(3,5-dihydroxystyryl)benzene-1,2-d...)
Affinity DataIC50: 4.70E+4nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50045936(CHEMBL69863 | 4-(3,5-dihydroxystyryl)benzene-1,2-d...)
Affinity DataIC50: 6.90E+4nMAssay Description:Inhibition of recombinant human liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553165(CHEMBL4754674)
Affinity DataIC50: 7.60E+4nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553165(CHEMBL4754674)
Affinity DataKi:  8.20E+4nMAssay Description:Mixed type inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553165(CHEMBL4754674)
Affinity DataKi:  8.20E+4nMAssay Description:Mixed type inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553165(CHEMBL4754674)
Affinity DataKi:  8.20E+4nMAssay Description:Mixed type inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553164(CHEMBL4741701)
Affinity DataIC50: 8.30E+4nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553165(CHEMBL4754674)
Affinity DataIC50: 8.90E+4nMAssay Description:Inhibition of recombinant human liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553157(CHEMBL440107)
Affinity DataIC50: 1.06E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553177(CHEMBL4742032)
Affinity DataIC50: 1.08E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM26188(1,2-Dihydroxybenzene, XI | CHEMBL280998 | benzene-...)
Affinity DataIC50: 1.23E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataIC50: 1.28E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM4375(3,4-Dihydroxycinnamate, XVII | cid_689043 | Caffei...)
Affinity DataIC50: 1.31E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50045936(CHEMBL69863 | 4-(3,5-dihydroxystyryl)benzene-1,2-d...)
Affinity DataKi:  1.36E+5nMAssay Description:Mixed type inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by Cornish-Bowden plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50045936(CHEMBL69863 | 4-(3,5-dihydroxystyryl)benzene-1,2-d...)
Affinity DataKi:  1.36E+5nMAssay Description:Mixed type inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50045936(CHEMBL69863 | 4-(3,5-dihydroxystyryl)benzene-1,2-d...)
Affinity DataKi:  1.36E+5nMAssay Description:Mixed type inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by Dixon plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553162(CHEMBL4798237)
Affinity DataIC50: 1.41E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553171(CHEMBL4794440)
Affinity DataIC50: 1.45E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553161(CHEMBL4757794)
Affinity DataIC50: 1.54E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553160(CHEMBL4791480)
Affinity DataIC50: 1.64E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553158(CHEMBL2009732)
Affinity DataIC50: 1.64E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553159(CHEMBL4764741)
Affinity DataIC50: 1.85E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553178(CHEMBL4756480)
Affinity DataIC50: 1.87E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553176(CHEMBL4597903)
Affinity DataIC50: 2.26E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553163(CHEMBL4741885)
Affinity DataIC50: 2.38E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM92758(3-Bromocatechol)
Affinity DataIC50: 2.74E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553175(CHEMBL4748612)
Affinity DataIC50: 2.77E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50242283(Methyl protocatechuate | methyl 3,4-dihydroxybenzo...)
Affinity DataIC50: 2.85E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553173(CHEMBL4750334)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553169(CHEMBL4794775)
Affinity DataIC50: 3.18E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553174(CHEMBL4780884)
Affinity DataIC50: 3.29E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553167(CHEMBL4793535)
Affinity DataIC50: 3.43E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50240171(CHEMBL3092389 | CHEBI:16971)
Affinity DataIC50: 3.60E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553168(CHEMBL4788184)
Affinity DataIC50: 3.62E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553170(CHEMBL4798533)
Affinity DataIC50: 3.67E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553172(CHEMBL4781582)
Affinity DataIC50: 3.89E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553166(CHEMBL4761488)
Affinity DataIC50: 4.67E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Bovine)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553156(CHEMBL4753152)
Affinity DataIC50: 4.78E+5nMAssay Description:Inhibition of recombinant bovine liver ARGI using L-arginine as substrate incubated for 60 mins by spectroscopic analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50553165(CHEMBL4754674)
Affinity DataIC50: 7.94E+5nMAssay Description:Inhibition of recombinant human ARG1 expressed in CHO-K1 cells assessed as reduction in urea level incubated for 24 hrs by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetArginase-1(Human)
Univ. Bourgogne Franche-Comt�

Curated by ChEMBL
LigandPNGBDBM50045936(CHEMBL69863 | 4-(3,5-dihydroxystyryl)benzene-1,2-d...)
Affinity DataIC50: 1.18E+6nMAssay Description:Inhibition of recombinant human ARG1 expressed in CHO-K1 cells assessed as reduction in urea level incubated for 24 hrs by colorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed