Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 50017963
TargetTyrosine-protein kinase receptor UFO(Human)
Oncowitan

Curated by ChEMBL
LigandPNGBDBM50606525(CHEMBL5218452)
Affinity DataIC50: 0.490nMAssay Description:Inhibition of AXL (unknown origin) by biochemical assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetAldo-keto reductase family 1 member C3(Human)
Oncowitan

Curated by ChEMBL
LigandPNGBDBM50051340(2-(2-Hydroxy-phenyl)-chroman-4-one | 2'-Hydroxyfla...)
Affinity DataIC50: 300nMAssay Description:Inhibition of human recombinant His-tagged AKR1C3 expressed in Escherichia coli BL21(DE3) incubated for 30 mins by HPLC analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Human)
Oncowitan

Curated by ChEMBL
LigandPNGBDBM50051340(2-(2-Hydroxy-phenyl)-chroman-4-one | 2'-Hydroxyfla...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human 11beta-HSD1 expressed in HEK-293 cells incubated for 10 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed