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Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50017961
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606516(CHEMBL5220372)
Affinity DataEC50:  0.930nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  0.0790nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606509(CHEMBL5220384)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606510(CHEMBL5219646)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606511(CHEMBL5219263)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606512(CHEMBL5218509)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606513(CHEMBL5220630)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606514(CHEMBL5220666)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606515(CHEMBL5219122)
Affinity DataEC50:  0.280nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606508(CHEMBL5220965)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606517(CHEMBL5221090)
Affinity DataEC50:  0.420nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606518(CHEMBL5219458)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606519(CHEMBL5220497)
Affinity DataEC50:  0.850nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606520(CHEMBL5218999)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606521(CHEMBL5220251)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606522(CHEMBL5219454)
Affinity DataEC50:  0.130nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606523(CHEMBL5218881)
Affinity DataEC50:  0.0980nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606524(CHEMBL5220241)
Affinity DataEC50:  0.280nMAssay Description:Agonist activity at human GCGR expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606516(CHEMBL5220372)
Affinity DataEC50:  0.620nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606509(CHEMBL5220384)
Affinity DataEC50:  0.160nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606510(CHEMBL5219646)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606511(CHEMBL5219263)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606512(CHEMBL5218509)
Affinity DataEC50:  0.560nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606513(CHEMBL5220630)
Affinity DataEC50:  0.730nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606514(CHEMBL5220666)
Affinity DataEC50:  0.680nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606515(CHEMBL5219122)
Affinity DataEC50:  0.0780nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606508(CHEMBL5220965)
Affinity DataEC50:  0.0410nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606517(CHEMBL5221090)
Affinity DataEC50:  0.570nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606518(CHEMBL5219458)
Affinity DataEC50:  0.450nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606519(CHEMBL5220497)
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606520(CHEMBL5218999)
Affinity DataEC50:  0.220nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606521(CHEMBL5220251)
Affinity DataEC50:  0.0530nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606522(CHEMBL5219454)
Affinity DataEC50:  0.0510nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606523(CHEMBL5218881)
Affinity DataEC50:  0.0310nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed
TargetGlucagon-like peptide 1 receptor(Human)
Affiliated Tumor Hospital of Guangxi Medical University

Curated by ChEMBL
LigandPNGBDBM50606524(CHEMBL5220241)
Affinity DataEC50:  0.0860nMAssay Description:Agonist activity at human GLP-1R expressed in HEK293 cells incubated for 30 mins and assessed as increase in cAMP accumulation measured by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2023
Entry Details
PubMed