Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50013456
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine

Curated by ChEMBL
LigandPNGBDBM50566090(CHEMBL4788526)
Affinity DataKd:  200nMAssay Description:Binding affinity to human RXRalpha-LBD assessed as binding constant from binding ratio at 327 nm by fluorometric titration assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine

Curated by ChEMBL
LigandPNGBDBM50566090(CHEMBL4788526)
Affinity DataKd:  257nMAssay Description:Binding affinity to human RXRalpha-LBD by fluorescence binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine

Curated by ChEMBL
LigandPNGBDBM50566090(CHEMBL4788526)
Affinity DataKi:  332nMAssay Description:Displacement of [3H]9cis-RA from human RXRalpha-LBD by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine

Curated by ChEMBL
LigandPNGBDBM50566089(CHEMBL4778155)
Affinity DataKi:  425nMAssay Description:Displacement of [3H]9cis-RA from human RXRalpha-LBD by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetRetinoic acid receptor RXR-alpha(Human)
Okayama University Graduate School of Medicine

Curated by ChEMBL
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataKi:  478nMAssay Description:Displacement of 6-(Ethyl-{5-isobutoxy-4-isopropyl-2-[(10-oxo-2,3,5,6-tetrahydro-1H,4H,10H-11-oxa-3a-aza-benzo[de]anthracene-9-carbonyl)-amino]-phenyl...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)