Compile Data Set for Download or QSAR
Report error Found 47 Enz. Inhib. hit(s) with all data for entry = 50013107
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562710(CHEMBL4759730)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50334252(3-(4-methylpiperazin-1-yl)-1-(phenylsulfonyl)-1H-i...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562696(CHEMBL4759208)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562703(CHEMBL4753562)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562710(CHEMBL4759730)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]-Raclopride from dopamine D2 receptor (unknown origin) incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562690(CHEMBL4795207)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 2A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562710(CHEMBL4759730)
Affinity DataKi:  41nMAssay Description:Binding affinity to 5-HT2A receptor (unknown origin) incubated for 1 hr by microbeta counting based displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562706(CHEMBL4744372)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562699(CHEMBL4763622)
Affinity DataKi:  82nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562716(CHEMBL4797942)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562695(CHEMBL4795614)
Affinity DataKi:  97nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562719(CHEMBL4753238)
Affinity DataKi:  108nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562711(CHEMBL4750481)
Affinity DataKi:  124nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562717(CHEMBL1501353)
Affinity DataKi:  127nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562707(CHEMBL4752848)
Affinity DataKi:  128nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562712(CHEMBL4743932)
Affinity DataKi:  146nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50187508(1-Benzenesulfonyl-1H-indole | 1-Phenylsulfonyl-1H-...)
Affinity DataKi:  159nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562705(CHEMBL4761081)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562710(CHEMBL4759730)
Affinity DataKi:  164nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-HT1A receptor (unknown origin) incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562691(CHEMBL4763575)
Affinity DataKi:  178nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562692(CHEMBL4740955)
Affinity DataKi:  211nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562714(CHEMBL4797400)
Affinity DataKi:  219nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562696(CHEMBL4759208)
Affinity DataKi:  241nMAssay Description:Displacement of [3H]-Raclopride from dopamine D2 receptor (unknown origin) incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562696(CHEMBL4759208)
Affinity DataKi:  247nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5-HT1A receptor (unknown origin) incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562718(CHEMBL4759121)
Affinity DataKi:  262nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562700(CHEMBL4753614)
Affinity DataKi:  360nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562693(CHEMBL4760297)
Affinity DataKi:  403nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562697(CHEMBL4763536)
Affinity DataKi:  409nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562713(CHEMBL4777921)
Affinity DataKi:  474nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562698(CHEMBL4764769)
Affinity DataKi:  558nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562709(CHEMBL4755749)
Affinity DataKi:  714nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562683(CHEMBL4752004)
Affinity DataKi:  1.15E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562694(CHEMBL4745715)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562704(CHEMBL4776760)
Affinity DataKi:  1.51E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562682(CHEMBL4783954)
Affinity DataKi:  1.66E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562708(CHEMBL4781626)
Affinity DataKi:  1.74E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562715(CHEMBL4746839)
Affinity DataKi:  2.03E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562681(CHEMBL4800552)
Affinity DataKi:  2.18E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562685(CHEMBL4747483)
Affinity DataKi:  2.56E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562680(CHEMBL4750657)
Affinity DataKi:  3.26E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562684(CHEMBL4753752)
Affinity DataKi:  4.05E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562689(CHEMBL4750554)
Affinity DataKi:  4.72E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562702(CHEMBL4742713)
Affinity DataKi:  4.85E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562686(CHEMBL4785319)
Affinity DataKi:  4.89E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562701(CHEMBL4759633)
Affinity DataKi:  5.25E+3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562687(CHEMBL4751913)
Affinity DataKi:  3.91E+4nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 6(Human)
Polish Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50562688(CHEMBL4751332)
Affinity DataKi:  4.99E+4nMAssay Description:Displacement of [3H]-LSD from human 5-HT6 receptor incubated for 1 hr by microbeta counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed