Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50012351
TargetApelin receptor(Rat)
Huazhong University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556824(CHEMBL4746142)
Affinity DataEC50:  8.80nMAssay Description:Agonist activity at APJ receptor in rat NRK-52E cells assessed as effect on cAMP accumulation incubated for 1 hr by cAMP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Huazhong University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556825(CHEMBL4787784)
Affinity DataEC50:  8nMAssay Description:Agonist activity at APJ receptor in rat NRK-52E cells assessed as effect on cAMP accumulation incubated for 1 hr by cAMP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Huazhong University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556826(CHEMBL4745863)
Affinity DataEC50:  6.90nMAssay Description:Agonist activity at APJ receptor in rat NRK-52E cells assessed as effect on cAMP accumulation incubated for 1 hr by cAMP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Huazhong University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556827(CHEMBL4748838)
Affinity DataEC50:  7.80nMAssay Description:Agonist activity at APJ receptor in rat NRK-52E cells assessed as effect on cAMP accumulation incubated for 1 hr by cAMP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetApelin receptor(Rat)
Huazhong University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556828(CHEMBL4798771)
Affinity DataEC50:  9.5nMAssay Description:Agonist activity at APJ receptor in rat NRK-52E cells assessed as effect on cAMP accumulation incubated for 1 hr by cAMP-Glo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Huazhong University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556826(CHEMBL4745863)
Affinity DataKi:  0.220nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Huazhong University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556827(CHEMBL4748838)
Affinity DataKi:  0.25nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Huazhong University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556825(CHEMBL4787784)
Affinity DataKi:  0.460nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Huazhong University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556828(CHEMBL4798771)
Affinity DataKi:  0.600nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Huazhong University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556824(CHEMBL4746142)
Affinity DataKi:  5.10nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed
TargetApelin receptor(Human)
Huazhong University of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556829(CHEMBL4743589)
Affinity DataKi:  5.60nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2022
Entry Details Article
PubMed