Compile Data Set for Download or QSAR
Report error Found 92 Enz. Inhib. hit(s) with all data for entry = 50012185
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555149(CHEMBL4746919)
Affinity DataEC50:  25nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555151(CHEMBL4740521)
Affinity DataEC50:  214nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555150(CHEMBL4793250)
Affinity DataEC50:  17nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555149(CHEMBL4746919)
Affinity DataEC50:  25nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555148(CHEMBL4745148)
Affinity DataEC50:  589nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555156(CHEMBL4750006)
Affinity DataEC50:  361nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555155(CHEMBL4788060)
Affinity DataEC50:  354nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555154(CHEMBL4800237)
Affinity DataEC50:  7.5nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555153(CHEMBL4744365)
Affinity DataEC50:  33nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555152(CHEMBL4761246)
Affinity DataEC50:  788nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555151(CHEMBL4740521)
Affinity DataEC50:  216nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555150(CHEMBL4793250)
Affinity DataEC50:  18nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555152(CHEMBL4761246)
Affinity DataEC50:  794nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555148(CHEMBL4745148)
Affinity DataEC50:  591nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555156(CHEMBL4750006)
Affinity DataEC50:  200nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555155(CHEMBL4788060)
Affinity DataEC50:  490nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555154(CHEMBL4800237)
Affinity DataEC50:  174nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555153(CHEMBL4744365)
Affinity DataEC50:  162nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555152(CHEMBL4761246)
Affinity DataEC50:  219nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555151(CHEMBL4740521)
Affinity DataEC50:  200nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555150(CHEMBL4793250)
Affinity DataEC50:  513nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555149(CHEMBL4746919)
Affinity DataEC50:  219nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555148(CHEMBL4745148)
Affinity DataEC50:  589nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555154(CHEMBL4800237)
Affinity DataEC50:  19nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555156(CHEMBL4750006)
Affinity DataEC50:  191nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555155(CHEMBL4788060)
Affinity DataEC50:  170nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555154(CHEMBL4800237)
Affinity DataEC50:  19nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555153(CHEMBL4744365)
Affinity DataEC50:  120nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555152(CHEMBL4761246)
Affinity DataEC50:  724nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555151(CHEMBL4740521)
Affinity DataEC50:  692nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555150(CHEMBL4793250)
Affinity DataEC50:  537nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555149(CHEMBL4746919)
Affinity DataEC50:  759nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555148(CHEMBL4745148)
Affinity DataEC50:  186nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555156(CHEMBL4750006)
Affinity DataEC50:  192nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555155(CHEMBL4788060)
Affinity DataEC50:  168nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetDelta-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555156(CHEMBL4750006)
Affinity DataEC50:  200nMAssay Description:Agonist activity at delta opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555153(CHEMBL4744365)
Affinity DataEC50:  120nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555152(CHEMBL4761246)
Affinity DataEC50:  719nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555151(CHEMBL4740521)
Affinity DataEC50:  697nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555150(CHEMBL4793250)
Affinity DataEC50:  532nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555149(CHEMBL4746919)
Affinity DataEC50:  752nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 2(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555148(CHEMBL4745148)
Affinity DataEC50:  185nMAssay Description:Agonist activity at NPFFR2 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555156(CHEMBL4750006)
Affinity DataEC50:  363nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555155(CHEMBL4788060)
Affinity DataEC50:  355nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555154(CHEMBL4800237)
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetNeuropeptide FF receptor 1(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555153(CHEMBL4744365)
Affinity DataEC50:  32nMAssay Description:Agonist activity at NPFFR1 (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMu-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555148(CHEMBL4745148)
Affinity DataEC50:  309nMAssay Description:Agonist activity at mu opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555154(CHEMBL4800237)
Affinity DataEC50:  871nMAssay Description:Agonist activity at kappa opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555155(CHEMBL4788060)
Affinity DataEC50:  741nMAssay Description:Agonist activity at kappa opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetKappa-type opioid receptor(Human)
Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50555156(CHEMBL4750006)
Affinity DataEC50:  2.46E+3nMAssay Description:Agonist activity at kappa opioid receptor (unknown origin) expressed in HEK293-A cells assessed as inhibition of forskolin-stimulated cAMP accumulati...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
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