Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50011607
TargetGastrin/cholecystokinin type B receptor(Human)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50024321(CHEMBL1328 | Peptavlon | ICI-50123 | 3-{2-[2-(3-te...)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at human CCK2R expressed in human A431 cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50549228(CHEMBL4758706)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human CCK2R expressed in human A431 cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50549227(CHEMBL4759105)
Affinity DataEC50:  14nMAssay Description:Agonist activity at human CCK2R expressed in human A431 cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50549226(CHEMBL4795913)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human CCK2R expressed in human A431 cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye ba...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50024321(CHEMBL1328 | Peptavlon | ICI-50123 | 3-{2-[2-(3-te...)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50549228(CHEMBL4758706)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50549227(CHEMBL4759105)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Rat)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50549226(CHEMBL4795913)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50549229(CHEMBL4761587)
Affinity DataIC50: 0.400nMAssay Description:Displacement of [125I][3-iodo Tyr12,Leu15]gastrin-I from human CCK2R expressed in human A431 cells measured after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50549227(CHEMBL4759105)
Affinity DataIC50: 0.600nMAssay Description:Displacement of [125I][3-iodo Tyr12,Leu15]gastrin-I from human CCK2R expressed in human A431 cells measured after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50549230(CHEMBL4795198)
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I][3-iodo Tyr12,Leu15]gastrin-I from human CCK2R expressed in human A431 cells measured after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50024321(CHEMBL1328 | Peptavlon | ICI-50123 | 3-{2-[2-(3-te...)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I][3-iodo Tyr12,Leu15]gastrin-I from human CCK2R expressed in human A431 cells measured after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50549228(CHEMBL4758706)
Affinity DataIC50: 1.30nMAssay Description:Displacement of [125I][3-iodo Tyr12,Leu15]gastrin-I from human CCK2R expressed in human A431 cells measured after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed
TargetGastrin/cholecystokinin type B receptor(Human)
Medical University of Innsbruck

Curated by ChEMBL
LigandPNGBDBM50549226(CHEMBL4795913)
Affinity DataIC50: 1.40nMAssay Description:Displacement of [125I][3-iodo Tyr12,Leu15]gastrin-I from human CCK2R expressed in human A431 cells measured after 1 hr by gamma counter analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2022
Entry Details Article
PubMed