Compile Data Set for Download or QSAR
Report error Found 22 Enz. Inhib. hit(s) with all data for entry = 50012132
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[2-(1H-indol-3-yl)-1-methylc...)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554436(CHEMBL4787709)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554435(CHEMBL4755394)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554423(CHEMBL4741966)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554422(CHEMBL4748728)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554437(CHEMBL4764498)
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554418(CHEMBL4787278)
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554429(CHEMBL4758924)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554421(CHEMBL4785870)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50287585(CHEMBL4169775)
Affinity DataIC50: 27nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554433(CHEMBL4741404)
Affinity DataIC50: 28nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554430(CHEMBL4764208)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554428(CHEMBL4742155)
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554419(CHEMBL4780646)
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554427(CHEMBL4757848)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554432(CHEMBL4745673)
Affinity DataIC50: 36nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554424(CHEMBL4784390)
Affinity DataIC50: 42nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554425(CHEMBL4745509)
Affinity DataIC50: 42nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554431(CHEMBL4763004)
Affinity DataIC50: 47nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554426(CHEMBL4759199)
Affinity DataIC50: 57nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554434(CHEMBL4765190)
Affinity DataIC50: 76nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMacrophage metalloelastase(Human)
University of California Riverside

Curated by ChEMBL
LigandPNGBDBM50554420(CHEMBL4788689)
Affinity DataIC50: 138nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly263 residues) expressed in Escherichia coli BL21 Codon Plus cells using 5-FAM/QX...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed