Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 50011387
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547574(CHEMBL4747964)
Affinity DataIC50: 3nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547568(CHEMBL4791554)
Affinity DataIC50: 3.10nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547569(CHEMBL4764193)
Affinity DataIC50: 3.40nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547572(CHEMBL4788971)
Affinity DataIC50: 3.60nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547573(CHEMBL4747827)
Affinity DataIC50: 4.20nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547571(CHEMBL4755277)
Affinity DataIC50: 4.70nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547566(CHEMBL4790062)
Affinity DataIC50: 4.80nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547567(CHEMBL4781886)
Affinity DataIC50: 4.80nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547575(CHEMBL4740349)
Affinity DataIC50: 7.40nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547565(CHEMBL4756743)
Affinity DataIC50: 7.5nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547516(CHEMBL4762897)
Affinity DataIC50: 10nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547550(CHEMBL4760303)
Affinity DataIC50: 11nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547560(CHEMBL4792032)
Affinity DataIC50: 11nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547515(CHEMBL4754176)
Affinity DataIC50: 13nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547555(CHEMBL4794133)
Affinity DataIC50: 16nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547576(CHEMBL4740544)
Affinity DataIC50: 17nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547514(CHEMBL4746924)
Affinity DataIC50: 19nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547562(CHEMBL4751630)
Affinity DataIC50: 20nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547563(CHEMBL4788462)
Affinity DataIC50: 24nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547570(CHEMBL4785277)
Affinity DataIC50: 26nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547561(CHEMBL4750320)
Affinity DataIC50: 30nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547552(CHEMBL4754751)
Affinity DataIC50: 34nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547551(CHEMBL4785587)
Affinity DataIC50: 44nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547548(CHEMBL4760005)
Affinity DataIC50: 55nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547559(CHEMBL4756985)
Affinity DataIC50: 55nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547513(CHEMBL4750619)
Affinity DataIC50: 55nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547512(CHEMBL4776337)
Affinity DataIC50: 70nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547510(CHEMBL4796106)
Affinity DataIC50: 91nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547553(CHEMBL4778658)
Affinity DataIC50: 91nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547564(CHEMBL4748504)
Affinity DataIC50: 101nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547558(CHEMBL4759189)
Affinity DataIC50: 107nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547511(CHEMBL4787250)
Affinity DataIC50: 115nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547508(CHEMBL4750670)
Affinity DataIC50: 166nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547556(CHEMBL4793109)
Affinity DataIC50: 180nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547529(CHEMBL4749322)
Affinity DataIC50: 192nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50006933(CHEMBL3134422)
Affinity DataIC50: 193nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547527(CHEMBL4747777)
Affinity DataIC50: 207nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547509(CHEMBL4752720)
Affinity DataIC50: 280nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547557(CHEMBL4743599)
Affinity DataIC50: 430nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547543(CHEMBL4778030)
Affinity DataIC50: 486nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547542(CHEMBL4777748)
Affinity DataIC50: 1.04E+3nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547544(CHEMBL4742010)
Affinity DataIC50: 1.59E+3nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547549(CHEMBL4786657)
Affinity DataIC50: 1.69E+3nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547530(CHEMBL4794380)
Affinity DataIC50: 1.77E+3nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547554(CHEMBL4762247)
Affinity DataIC50: 4.03E+3nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547546(CHEMBL4793306)
Affinity DataIC50: 4.30E+3nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547526(CHEMBL4779152)
Affinity DataIC50: 4.57E+3nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50540624(CHEMBL4647979)
Affinity DataIC50: 5.88E+3nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547541(CHEMBL4779325)
Affinity DataIC50: 6.06E+3nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetKelch-like ECH-associated protein 1(Human)
Irbm

Curated by ChEMBL
LigandPNGBDBM50547534(CHEMBL4752836)
Affinity DataIC50: 6.08E+3nMAssay Description:Binding affinity to human KEAP1 Kelch domain (322 to 609 residues) incubated for 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
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