Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50012109
TargetG protein-coupled receptor kinase 5(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554263(CHEMBL4740635)
Affinity DataKd:  3.43E+4nMAssay Description:Binding affinity to GRK5 (unknown origin) by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 5(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554262(CHEMBL4791786)
Affinity DataKd: >8.33E+4nMAssay Description:Binding affinity to GRK5 (unknown origin) by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 5(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554261(CHEMBL4742242)
Affinity DataKd: >8.33E+4nMAssay Description:Binding affinity to GRK5 (unknown origin) by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554259(CHEMBL4788026)
Affinity DataKd:  3.33E+3nMAssay Description:Binding affinity to full length human GRK2 by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM22416(PAROXETINE | CHEMBL490 | (3S,4R)-3-[(1,3-benzodiox...)
Affinity DataKd:  2.98E+3nMAssay Description:Binding affinity to full length human GRK2 by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50173313(CHEMBL1738878)
Affinity DataKd:  2nMAssay Description:Binding affinity to full length human GRK2 by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 5(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554260(CHEMBL4776422)
Affinity DataKd: >8.33E+4nMAssay Description:Binding affinity to GRK5 (unknown origin) by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 5(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554259(CHEMBL4788026)
Affinity DataKd: >8.33E+4nMAssay Description:Binding affinity to GRK5 (unknown origin) by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRhodopsin kinase GRK1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554263(CHEMBL4740635)
Affinity DataKd:  1.45E+4nMAssay Description:Binding affinity to GRK1 (unknown origin) by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRhodopsin kinase GRK1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554262(CHEMBL4791786)
Affinity DataKd: >8.33E+4nMAssay Description:Binding affinity to GRK1 (unknown origin) by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRhodopsin kinase GRK1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554261(CHEMBL4742242)
Affinity DataKd: >8.33E+4nMAssay Description:Binding affinity to GRK1 (unknown origin) by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRhodopsin kinase GRK1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554260(CHEMBL4776422)
Affinity DataKd: >8.33E+4nMAssay Description:Binding affinity to GRK1 (unknown origin) by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRhodopsin kinase GRK1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554259(CHEMBL4788026)
Affinity DataKd:  4.76E+4nMAssay Description:Binding affinity to GRK1 (unknown origin) by Thermofluor thermal shift assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554257(CHEMBL4742990)
Affinity DataIC50: 6nMAssay Description:Inhibition of human GRK2 by LANCE assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554266(CHEMBL4785990)
Affinity DataIC50: 9nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554267(CHEMBL4760734)
Affinity DataIC50: 10nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554268(CHEMBL4745381)
Affinity DataIC50: 10nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554257(CHEMBL4742990)
Affinity DataIC50: 11nMAssay Description:Inhibition of human Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554276(CHEMBL4753687)
Affinity DataIC50: 12nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554274(CHEMBL4782910)
Affinity DataIC50: 13nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554272(CHEMBL4751285)
Affinity DataIC50: 18nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 19nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554270(CHEMBL4752236)
Affinity DataIC50: 78nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554263(CHEMBL4740635)
Affinity DataIC50: 95nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 137nMAssay Description:Inhibition of human Aurora AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554271(CHEMBL4782250)
Affinity DataIC50: 206nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554257(CHEMBL4742990)
Affinity DataIC50: 246nMAssay Description:Inhibition of human ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554264(CHEMBL4755199)
Affinity DataIC50: 278nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554265(CHEMBL4793755)
Affinity DataIC50: 472nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554257(CHEMBL4742990)
Affinity DataIC50: 483nMAssay Description:Inhibition of RSK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRho-associated protein kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 1.27E+3nMAssay Description:Inhibition of human ROCK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554257(CHEMBL4742990)
Affinity DataIC50: 1.45E+3nMAssay Description:Inhibition of human PKBalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554275(CHEMBL4762347)
Affinity DataIC50: 2.11E+3nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554273(CHEMBL4783892)
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRibosomal protein S6 kinase alpha-1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 3.15E+3nMAssay Description:Inhibition of RSK1 (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554257(CHEMBL4742990)
Affinity DataIC50: 3.27E+3nMAssay Description:Inhibition of human GRK6More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCalcium/calmodulin-dependent protein kinase type II subunit beta(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554257(CHEMBL4742990)
Affinity DataIC50: 3.85E+3nMAssay Description:Inhibition of human CaMK2betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBeta-adrenergic receptor kinase 1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554259(CHEMBL4788026)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human GRK2 by transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 5(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554257(CHEMBL4742990)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of human GRK5More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554257(CHEMBL4742990)
Affinity DataIC50: 9.07E+3nMAssay Description:Inhibition of human PKCbeta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRhodopsin kinase GRK7(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554257(CHEMBL4742990)
Affinity DataIC50: 9.14E+3nMAssay Description:Inhibition of human GRK7More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein kinase C alpha type(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human PKCalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCalcium/calmodulin-dependent protein kinase type II subunit beta(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human CaMK2betaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetProtein kinase C beta type(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human PKCbeta1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRhodopsin kinase GRK7(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human GRK7More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 6(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human GRK6More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetG protein-coupled receptor kinase 5(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human GRK5More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRhodopsin kinase GRK1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human GRK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRhodopsin kinase GRK1(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554257(CHEMBL4742990)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human GRK1More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50554258(CHEMBL4744858)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human PKBalphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
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