Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50012100
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Human)
The Chinese University of Hong Kong (Shenzhen)

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50: 179nMAssay Description:Inhibition of GST-tagged recombinant human full length MNK1 expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
The Chinese University of Hong Kong (Shenzhen)

Curated by ChEMBL
LigandPNGBDBM50049395(5,7-dihydroxy-2-(4-hydroxyphenyl)-6-methoxy-4H-chr...)
Affinity DataIC50: 252nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length MNK2 expressed in baculovirus expression system incubated for 1 hr by Kinase Tracer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
The Chinese University of Hong Kong (Shenzhen)

Curated by ChEMBL
LigandPNGBDBM7458(Naringenin, 18 | 5,7-dihydroxy-2-(4-hydroxyphenyl)...)
Affinity DataIC50: 308nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length MNK2 expressed in baculovirus expression system incubated for 1 hr by Kinase Tracer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
The Chinese University of Hong Kong (Shenzhen)

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataIC50: 579nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length MNK2 expressed in baculovirus expression system incubated for 1 hr by Kinase Tracer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
The Chinese University of Hong Kong (Shenzhen)

Curated by ChEMBL
LigandPNGBDBM50187658(7-O-methylapigenin | genkwanin | 5-hydroxy-2-(4-hy...)
Affinity DataIC50: 979nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length MNK2 expressed in baculovirus expression system incubated for 1 hr by Kinase Tracer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 1(Human)
The Chinese University of Hong Kong (Shenzhen)

Curated by ChEMBL
LigandPNGBDBM50049395(5,7-dihydroxy-2-(4-hydroxyphenyl)-6-methoxy-4H-chr...)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of GST-tagged recombinant human full length MNK1 expressed in insect cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
The Chinese University of Hong Kong (Shenzhen)

Curated by ChEMBL
LigandPNGBDBM50554183(CHEBI:75162 | CHEMBL77588)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length MNK2 expressed in baculovirus expression system incubated for 1 hr by Kinase Tracer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
The Chinese University of Hong Kong (Shenzhen)

Curated by ChEMBL
LigandPNGBDBM50554187(CHEMBL4097277)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length MNK2 expressed in baculovirus expression system incubated for 1 hr by Kinase Tracer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
The Chinese University of Hong Kong (Shenzhen)

Curated by ChEMBL
LigandPNGBDBM50554186(CHEMBL4747606)
Affinity DataIC50: 4.67E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length MNK2 expressed in baculovirus expression system incubated for 1 hr by Kinase Tracer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
The Chinese University of Hong Kong (Shenzhen)

Curated by ChEMBL
LigandPNGBDBM50554185(CHEMBL4740978)
Affinity DataIC50: 6.49E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length MNK2 expressed in baculovirus expression system incubated for 1 hr by Kinase Tracer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetMAP kinase-interacting serine/threonine-protein kinase 2(Human)
The Chinese University of Hong Kong (Shenzhen)

Curated by ChEMBL
LigandPNGBDBM50554184(CHEMBL4755408)
Affinity DataIC50: 8.26E+3nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human full length MNK2 expressed in baculovirus expression system incubated for 1 hr by Kinase Tracer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed