Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 50018380
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607924(CHEMBL5278864)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of JAK3 (unknown origin) incubated for 45 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50501537(CHEMBL4085582)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 1 hr followed by substrate addition and measured after 1 hr by Z-lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607926(CHEMBL5270127)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 1 hr followed by substrate addition and measured after 1 hr by Z-lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607927(CHEMBL5272677)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 1 hr followed by substrate addition and measured after 1 hr by Z-lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607924(CHEMBL5278864)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 1 hr followed by substrate addition and measured after 1 hr by Z-lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607926(CHEMBL5270127)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of JAK3 (unknown origin) incubated for 45 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50501537(CHEMBL4085582)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of JAK3 (unknown origin) incubated for 45 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607927(CHEMBL5272677)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of JAK3 (unknown origin) incubated for 45 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50501537(CHEMBL4085582)
Affinity DataIC50: 0.770nMAssay Description:Inhibition of JAK3 (unknown origin) incubated for 45 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607926(CHEMBL5270127)
Affinity DataIC50: 1nMAssay Description:Inhibition of JAK3 (unknown origin) incubated for 45 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607927(CHEMBL5272677)
Affinity DataIC50: 11nMAssay Description:Inhibition of JAK3 (unknown origin) incubated for 45 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607924(CHEMBL5278864)
Affinity DataIC50: 26nMAssay Description:Inhibition of MELK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607924(CHEMBL5278864)
Affinity DataIC50: 56nMAssay Description:Inhibition of JAK3 (unknown origin) incubated for 45 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607925(CHEMBL5270221)
Affinity DataIC50: 56nMAssay Description:Inhibition of JAK3 (unknown origin) incubated for 45 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetMaternal embryonic leucine zipper kinase(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607928(CHEMBL5287531)
Affinity DataIC50: 222nMAssay Description:Inhibition of MELK (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetDual specificity mitogen-activated protein kinase kinase 4(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607924(CHEMBL5278864)
Affinity DataIC50: 281nMAssay Description:Inhibition of MAP2K4 (unknown origin) at 100 uM preincubated for 1 hr followed by substrate addition and measured after 1 hr by Z-lyte assay relative...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607925(CHEMBL5270221)
Affinity DataIC50: 399nMAssay Description:Inhibition of RSK2 (unknown origin) at 100 uM preincubated for 1 hr followed by substrate addition and measured after 1 hr by Z-lyte assay relative t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetRibosomal protein S6 kinase alpha-3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607924(CHEMBL5278864)
Affinity DataIC50: 399nMAssay Description:Inhibition of RSK2 (unknown origin) at 100 uM preincubated for 1 hr followed by substrate addition and measured after 1 hr by Z-lyte assay relative t...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607928(CHEMBL5287531)
Affinity DataIC50: 832nMAssay Description:Inhibition of JAK3 (unknown origin) preincubated for 1 hr followed by substrate addition and measured after 1 hr by Z-lyte assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Research Centre For Natural Sciences

Curated by ChEMBL
LigandPNGBDBM50607928(CHEMBL5287531)
Affinity DataIC50: 832nMAssay Description:Inhibition of JAK3 (unknown origin) incubated for 45 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed