Compile Data Set for Download or QSAR
Report error Found 128 Enz. Inhib. hit(s) with all data for entry = 50011550
LigandChemical structure of BindingDB Monomer ID 50369965BDBM50369965(Cetrotide | CETRORELIX)
Affinity DataKd:  0.00200nMAssay Description:Inhibition of Tag-lite green-labeled agonist binding to terbium fluorophore-labeled human N-terminal SNAP-tag GnRh receptor expressed in HEK293 cells...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50369965BDBM50369965(Cetrotide | CETRORELIX)
Affinity DataKd:  0.135nMAssay Description:Inhibition of Tag-lite green-labeled agonist binding to terbium fluorophore-labeled human N-terminal SNAP-tag GnRh receptor expressed in HEK293 cells...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347982BDBM50347982(CHEMBL1800159 | US20250000864, Compound Relugolix)
Affinity DataKd:  0.372nMAssay Description:Inhibition of Tag-lite green-labeled agonist binding to terbium fluorophore-labeled human N-terminal SNAP-tag GnRh receptor expressed in HEK293 cells...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50347982BDBM50347982(CHEMBL1800159 | US20250000864, Compound Relugolix)
Affinity DataKd:  0.840nMAssay Description:Inhibition of Tag-lite green-labeled agonist binding to terbium fluorophore-labeled human N-terminal SNAP-tag GnRh receptor expressed in HEK293 cells...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50274930BDBM50274930((R)-4-{2-[5-(2-Fluoro-3-methoxyphenyl)-3-(2-fluoro...)
Affinity DataKd:  1.20nMAssay Description:Inhibition of Tag-lite green-labeled agonist binding to terbium fluorophore-labeled human N-terminal SNAP-tag GnRh receptor expressed in HEK293 cells...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50274930BDBM50274930((R)-4-{2-[5-(2-Fluoro-3-methoxyphenyl)-3-(2-fluoro...)
Affinity DataKd:  3.20nMAssay Description:Inhibition of Tag-lite green-labeled agonist binding to terbium fluorophore-labeled human N-terminal SNAP-tag GnRh receptor expressed in HEK293 cells...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548493BDBM50548493(BAY-784)
Affinity DataKd:  5.5nMAssay Description:Inhibition of Tag-lite green-labeled agonist binding to terbium fluorophore-labeled human N-terminal SNAP-tag GnRh receptor expressed in HEK293 cells...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548493BDBM50548493(BAY-784)
Affinity DataKd:  9.80nMAssay Description:Inhibition of Tag-lite green-labeled agonist binding to terbium fluorophore-labeled human N-terminal SNAP-tag GnRh receptor expressed in HEK293 cells...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548475BDBM50548475(CHEMBL4747248)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548486BDBM50548486(CHEMBL4741994)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548470BDBM50548470(CHEMBL4749974)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548470BDBM50548470(CHEMBL4749974)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548472BDBM50548472(CHEMBL4749790)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548472BDBM50548472(CHEMBL4749790)
Affinity DataIC50: 15nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50041550BDBM50041550(CHEMBL3358413)
Affinity DataIC50: 16nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548469BDBM50548469(CHEMBL4762368)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548475BDBM50548475(CHEMBL4747248)
Affinity DataIC50: 18nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548468BDBM50548468(CHEMBL4747322)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548463BDBM50548463(CHEMBL4781434)
Affinity DataIC50: 20nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548493BDBM50548493(BAY-784)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548488BDBM50548488(CHEMBL4780737)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548488BDBM50548488(CHEMBL4780737)
Affinity DataIC50: 21nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548486BDBM50548486(CHEMBL4741994)
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548483BDBM50548483(CHEMBL4761024)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548493BDBM50548493(BAY-784)
Affinity DataIC50: 24nMAssay Description:Antagonist activity at rat GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548470BDBM50548470(CHEMBL4749974)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548467BDBM50548467(CHEMBL4787856)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548470BDBM50548470(CHEMBL4749974)
Affinity DataIC50: 26nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548493BDBM50548493(BAY-784)
Affinity DataIC50: 27nMAssay Description:Inhibition of Tag-lite green-labeled agonist binding to terbium fluorophore-labeled human N-terminal SNAP-tag GnRh receptor expressed in HEK293 cells...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548473BDBM50548473(CHEMBL4740373)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at rat GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548473BDBM50548473(CHEMBL4740373)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at rat GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548472BDBM50548472(CHEMBL4749790)
Affinity DataIC50: 28nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548472BDBM50548472(CHEMBL4749790)
Affinity DataIC50: 28nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548472BDBM50548472(CHEMBL4749790)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at rat GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548472BDBM50548472(CHEMBL4749790)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at rat GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548474BDBM50548474(CHEMBL4779806)
Affinity DataIC50: 34nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548471BDBM50548471(CHEMBL4782228)
Affinity DataIC50: 35nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548469BDBM50548469(CHEMBL4762368)
Affinity DataIC50: 36nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548478BDBM50548478(CHEMBL4746174)
Affinity DataIC50: 38nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548458BDBM50548458(CHEMBL4756920)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at rat GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548458BDBM50548458(CHEMBL4756920)
Affinity DataIC50: 40nMAssay Description:Antagonist activity at rat GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followed ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548468BDBM50548468(CHEMBL4747322)
Affinity DataIC50: 45nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548483BDBM50548483(CHEMBL4761024)
Affinity DataIC50: 47nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548465BDBM50548465(CHEMBL4745391)
Affinity DataIC50: 48nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548484BDBM50548484(CHEMBL4740379)
Affinity DataIC50: 53nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548464BDBM50548464(CHEMBL4793643)
Affinity DataIC50: 53nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50041550BDBM50041550(CHEMBL3358413)
Affinity DataIC50: 54nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of buserelin-induced response preincubated for 20 mins fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548471BDBM50548471(CHEMBL4782228)
Affinity DataIC50: 54nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548477BDBM50548477(CHEMBL4760799)
Affinity DataIC50: 56nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50548458BDBM50548458(CHEMBL4756920)
Affinity DataIC50: 60nMAssay Description:Antagonist activity at human GnRH receptor expressed in CHO-K1 cells assessed as inhibition of LHRH-induced response preincubated for 20 mins followe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
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