Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 50010922
TargetProprotein convertase subtilisin/kexin type 9(Human)
Lauren Mccallister

Curated by ChEMBL
LigandPNGBDBM50543439(CHEMBL4642977)
Affinity DataIC50: 0.152nMAssay Description:Inhibition of human PCSK9 by Alexa Fluor 647 staining based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 9(Human)
Lauren Mccallister

Curated by ChEMBL
LigandPNGBDBM50543440(CHEMBL4635142)
Affinity DataIC50: 0.327nMAssay Description:Inhibition of human PCSK9 by Alexa Fluor 647 staining based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 9(Human)
Lauren Mccallister

Curated by ChEMBL
LigandPNGBDBM50543441(CHEMBL4642595)
Affinity DataIC50: 0.438nMAssay Description:Inhibition of human PCSK9 by Alexa Fluor 647 staining based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 9(Human)
Lauren Mccallister

Curated by ChEMBL
LigandPNGBDBM50543444(CHEMBL4641251)
Affinity DataIC50: 0.570nMAssay Description:Inhibition of human PCSK9 by Alexa Fluor 647 staining based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 9(Human)
Lauren Mccallister

Curated by ChEMBL
LigandPNGBDBM50543442(CHEMBL4645450)
Affinity DataIC50: 0.850nMAssay Description:Inhibition of human PCSK9 by Alexa Fluor 647 staining based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed
TargetProprotein convertase subtilisin/kexin type 9(Human)
Lauren Mccallister

Curated by ChEMBL
LigandPNGBDBM50543443(CHEMBL4638184)
Affinity DataIC50: 0.930nMAssay Description:Inhibition of human PCSK9 by Alexa Fluor 647 staining based TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/13/2021
Entry Details Article
PubMed