Compile Data Set for Download or QSAR
Report error Found 15 Enz. Inhib. hit(s) with all data for entry = 50011346
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547296BDBM50547296(CHEMBL4761521)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase C(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381716BDBM50381716(US8722890, 1 | US8722890, 2 | ABT-348 | ILORASERTI...)
Affinity DataIC50: 7nMAssay Description:Inhibition of AuroraC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381716BDBM50381716(US8722890, 1 | US8722890, 2 | ABT-348 | ILORASERTI...)
Affinity DataIC50: 12nMAssay Description:Inhibition of AuroraB (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50004205BDBM50004205(MK-0457 | MK-045 | VX-680 | VX-68 | TOZASERTIB | U...)
Affinity DataIC50: 15nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547295BDBM50547295(CHEMBL4763465)
Affinity DataIC50: 21nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547300BDBM50547300(CHEMBL4790560)
Affinity DataIC50: 42nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547301BDBM50547301(CHEMBL4744828)
Affinity DataIC50: 68nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase A(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50381716BDBM50381716(US8722890, 1 | US8722890, 2 | ABT-348 | ILORASERTI...)
Affinity DataIC50: 120nMAssay Description:Inhibition of AuroraA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547294BDBM50547294(CHEMBL4755343)
Affinity DataIC50: 142nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547298BDBM50547298(CHEMBL4761439)
Affinity DataIC50: 206nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547293BDBM50547293(CHEMBL4758452)
Affinity DataIC50: 282nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547291BDBM50547291(CHEMBL4794671)
Affinity DataIC50: 294nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547297BDBM50547297(CHEMBL4745882)
Affinity DataIC50: 295nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547292BDBM50547292(CHEMBL4795345)
Affinity DataIC50: 360nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetAurora kinase B(Human)
Lanzhou University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50547299BDBM50547299(CHEMBL4784626)
Affinity DataIC50: 364nMAssay Description:Inhibition of AuroraB (unknown origin) by Kinase-Glo luminescent kinase assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed