Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50011548
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548442BDBM50548442(CHEMBL4754678)
Affinity DataKi:  16nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548446BDBM50548446(CHEMBL4792331)
Affinity DataKi:  40nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548441BDBM50548441(CHEMBL4786474)
Affinity DataKi:  41nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548444BDBM50548444(CHEMBL4745679)
Affinity DataKi:  42nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548440BDBM50548440(CHEMBL4790325)
Affinity DataKi:  46nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548450BDBM50548450(CHEMBL4749809)
Affinity DataKi:  60nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548445BDBM50548445(CHEMBL4794916)
Affinity DataKi:  60nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548452BDBM50548452(CHEMBL4795214)
Affinity DataKi:  66nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548447BDBM50548447(CHEMBL4759843)
Affinity DataKi:  110nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548444BDBM50548444(CHEMBL4745679)
Affinity DataKi:  130nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548455BDBM50548455(CHEMBL4744226)
Affinity DataKi:  130nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548443BDBM50548443(CHEMBL4778448)
Affinity DataKi:  143nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548453BDBM50548453(CHEMBL4787083)
Affinity DataKi:  176nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548442BDBM50548442(CHEMBL4754678)
Affinity DataKi:  230nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548445BDBM50548445(CHEMBL4794916)
Affinity DataKi:  270nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548455BDBM50548455(CHEMBL4744226)
Affinity DataKi:  290nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548441BDBM50548441(CHEMBL4786474)
Affinity DataKi:  340nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548447BDBM50548447(CHEMBL4759843)
Affinity DataKi:  350nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548440BDBM50548440(CHEMBL4790325)
Affinity DataKi:  350nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548446BDBM50548446(CHEMBL4792331)
Affinity DataKi:  400nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548452BDBM50548452(CHEMBL4795214)
Affinity DataKi:  460nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548454BDBM50548454(CHEMBL4762562)
Affinity DataKi:  480nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548454BDBM50548454(CHEMBL4762562)
Affinity DataKi:  550nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548451BDBM50548451(CHEMBL4787392)
Affinity DataKi:  570nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548456BDBM50548456(CHEMBL4760324)
Affinity DataKi:  800nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548453BDBM50548453(CHEMBL4787083)
Affinity DataKi:  870nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548448BDBM50548448(CHEMBL4758401)
Affinity DataKi:  870nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Human)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548451BDBM50548451(CHEMBL4787392)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of human IMPDH2 expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548449BDBM50548449(CHEMBL4796033)
Affinity DataKi:  1.70E+3nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed
TargetInosine-5'-monophosphate dehydrogenase(Cryptosporidium parvum)
University of Houston

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50548456BDBM50548456(CHEMBL4760324)
Affinity DataKi:  2.80E+3nMAssay Description:Inhibition of Cryptosporidium parvum IMPDH expressed in Escherichia coli assessed as apparent inhibition constant using NAD as substrate by fluoresce...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2022
Entry Details Article
PubMed