Compile Data Set for Download or QSAR
Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50012049
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553559(CHEMBL4795699)
Affinity DataKd:  2.54E+4nMAssay Description:Binding affinity to CBP BRD (unknown origin) by microscale thermophoresis assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553559(CHEMBL4795699)
Affinity DataIC50: 20nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553573(CHEMBL4790542)
Affinity DataIC50: 37nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553574(CHEMBL4741233)
Affinity DataIC50: 40nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553563(CHEMBL4793642)
Affinity DataIC50: 46nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553572(CHEMBL4791519)
Affinity DataIC50: 48nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553576(CHEMBL4776578)
Affinity DataIC50: 52nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553570(CHEMBL4779896)
Affinity DataIC50: 54nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553562(CHEMBL4783664)
Affinity DataIC50: 55nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553555(CHEMBL4758366)
Affinity DataIC50: 63nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553578(CHEMBL4784945)
Affinity DataIC50: 74nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553566(CHEMBL4755549)
Affinity DataIC50: 77nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553575(CHEMBL4778341)
Affinity DataIC50: 85nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553571(CHEMBL4756910)
Affinity DataIC50: 89nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553560(CHEMBL4743523)
Affinity DataIC50: 91nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553561(CHEMBL4792407)
Affinity DataIC50: 93nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553577(CHEMBL4791402)
Affinity DataIC50: 93nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553567(CHEMBL4740324)
Affinity DataIC50: 95nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553569(CHEMBL4755792)
Affinity DataIC50: 102nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553565(CHEMBL4783911)
Affinity DataIC50: 103nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553568(CHEMBL4776036)
Affinity DataIC50: 195nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553555(CHEMBL4758366)
Affinity DataIC50: 213nMAssay Description:Inhibition of GST-tagged CBP BRD (unknown origin) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553564(CHEMBL4780426)
Affinity DataIC50: 286nMAssay Description:Inhibition of CBP BRD (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553558(CHEMBL4760515)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of GST-tagged CBP BRD (unknown origin) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553556(CHEMBL4780221)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of GST-tagged CBP BRD (unknown origin) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553559(CHEMBL4795699)
Affinity DataIC50: 8.40E+3nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by ALPHAScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50178219(CHEMBL3814752)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of BRD4 BD1 (unknown origin) by ALPHAScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50178219(CHEMBL3814752)
Affinity DataIC50: 1.88E+4nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by ALPHAScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetBromodomain-containing protein 4(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553559(CHEMBL4795699)
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of BRD4 BD2 (unknown origin) by ALPHAScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed
TargetCREB-binding protein(Human)
Chinese Academy of Sciences

Curated by ChEMBL
LigandPNGBDBM50553557(CHEMBL4762596)
Affinity DataIC50: 6.33E+4nMAssay Description:Inhibition of GST-tagged CBP BRD (unknown origin) incubated for 30 mins by HTRF assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2022
Entry Details Article
PubMed