Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50013407
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565572(CHEMBL4800688)
Affinity DataIC50: 0.508nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565556(CHEMBL4787929)
Affinity DataIC50: 0.508nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565559(CHEMBL4792017)
Affinity DataIC50: 0.508nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565570(CHEMBL4798376)
Affinity DataIC50: 0.508nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565569(CHEMBL4780069)
Affinity DataIC50: 0.508nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565571(CHEMBL4790038)
Affinity DataIC50: 0.577nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565558(CHEMBL4783888)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565583(CHEMBL4780169)
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565555(CHEMBL4795375)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565586(CHEMBL4799529)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565585(CHEMBL4776291)
Affinity DataIC50: 2.20nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50402023(BI 6727 | VOLASERTIB)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565577(CHEMBL4784741)
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565573(CHEMBL4785567)
Affinity DataIC50: 3.30nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565582(CHEMBL4790028)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565564(CHEMBL4784781)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565576(CHEMBL4779654)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565581(CHEMBL4800085)
Affinity DataIC50: 4.30nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565557(CHEMBL4800017)
Affinity DataIC50: 4.40nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565574(CHEMBL4783122)
Affinity DataIC50: 4.60nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565552(CHEMBL4787496)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565584(CHEMBL4778470)
Affinity DataIC50: 4.70nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565575(CHEMBL4778422)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565565(CHEMBL4796797)
Affinity DataIC50: 5nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565561(CHEMBL4799183)
Affinity DataIC50: 5.10nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565562(CHEMBL4790807)
Affinity DataIC50: 5.30nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565554(CHEMBL4776345)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565563(CHEMBL4781522)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565553(CHEMBL4783750)
Affinity DataIC50: 8.10nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565578(CHEMBL4793797)
Affinity DataIC50: 29nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565579(CHEMBL4777642)
Affinity DataIC50: 50nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565580(CHEMBL4800439)
Affinity DataIC50: 189nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565566(CHEMBL4793185)
Affinity DataIC50: 219nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565567(CHEMBL4777753)
Affinity DataIC50: 3.51E+3nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565560(CHEMBL4780899)
Affinity DataIC50: 4.18E+3nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetSerine/threonine-protein kinase PLK1(Human)
Xiamen University

Curated by ChEMBL
LigandPNGBDBM50565568(CHEMBL4799010)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of human PLK1 using casein as substrate in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed