Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50013403
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
University of W£Rzburg
Curated by ChEMBL
University of W£Rzburg
Curated by ChEMBL
Affinity DataKd: 800nMAssay Description:Binding affinity to Pin1 (unknown origin) preincubated for 2 hrs followed by UV irradiation for 15 mins by SDS-PAGE gel based photoaffinity labelling...More data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Inhibition of human FKBP12 assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubated for 4 mins b...More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of human FKBP12 assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubated for 4 mins b...More data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of human FKBP12 assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubated for 4 mins b...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human FKBP12 assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubated for 4 mins b...More data for this Ligand-Target Pair
TargetPeptidyl-prolyl cis-trans isomerase NIMA-interacting 1(Human)
University of W£Rzburg
Curated by ChEMBL
University of W£Rzburg
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of human Pin1 assessed as reduction in PPIase activity using Suc-Ala-Glu-Pro-Phe-MCA as substrate measured for 20 secs by fluorescence met...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of Legionella pneumophila Mip assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of Legionella pneumophila Mip assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of Legionella pneumophila Mip assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 2.18E+4nMAssay Description:Inhibition of Legionella pneumophila Mip assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 3.17E+4nMAssay Description:Inhibition of Legionella pneumophila Mip assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubate...More data for this Ligand-Target Pair
Affinity DataIC50: 3.61E+4nMAssay Description:Inhibition of human FKBP12 assessed as reduction in PPIase activity using succinyl-Ala-Leu-Pro-Phe-4-nitroanilide as substrate incubated for 4 mins b...More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibition of recombinant human FKBP12 expressed in Escherichia coli using succinyl-Ala-Phe-Pro-Phe-4-nitroanilide as substrateMore data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Inhibition of recombinant human FKBP12 expressed in Escherichia coli using succinyl-Ala-Phe-Pro-Phe-4-nitroanilide as substrateMore data for this Ligand-Target Pair
