Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 50013397
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565488(CHEMBL4783386)
Affinity DataIC50: 400nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM25737(12-[(adamantan-1-ylcarbamoyl)amino]dodecanoic acid...)
Affinity DataIC50: 490nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565490(CHEMBL4788670)
Affinity DataIC50: 550nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 950nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565489(CHEMBL4779788)
Affinity DataIC50: 980nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565483(CHEMBL4790503)
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565494(CHEMBL4799379)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565488(CHEMBL4783386)
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565486(CHEMBL4789344)
Affinity DataIC50: 1.57E+3nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565493(CHEMBL4799227)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565487(CHEMBL4790061)
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565491(CHEMBL4789520)
Affinity DataIC50: 1.84E+3nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565490(CHEMBL4788670)
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565485(CHEMBL4792522)
Affinity DataIC50: 1.99E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565489(CHEMBL4779788)
Affinity DataIC50: 2.03E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565494(CHEMBL4799379)
Affinity DataIC50: 2.05E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565483(CHEMBL4790503)
Affinity DataIC50: 2.15E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565486(CHEMBL4789344)
Affinity DataIC50: 2.18E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565484(CHEMBL4777518)
Affinity DataIC50: 2.38E+3nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565484(CHEMBL4777518)
Affinity DataIC50: 2.48E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565487(CHEMBL4790061)
Affinity DataIC50: 2.89E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565492(CHEMBL4794910)
Affinity DataIC50: 3.04E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565492(CHEMBL4794910)
Affinity DataIC50: 3.31E+3nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565491(CHEMBL4789520)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565485(CHEMBL4792522)
Affinity DataIC50: 4.01E+3nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565493(CHEMBL4799227)
Affinity DataIC50: 4.12E+3nMAssay Description:Inhibition of recombinant human COX2 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 6.12E+3nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565488(CHEMBL4783386)
Affinity DataIC50: 8.72E+3nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565483(CHEMBL4790503)
Affinity DataIC50: 8.99E+3nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565494(CHEMBL4799379)
Affinity DataIC50: 9.12E+3nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565485(CHEMBL4792522)
Affinity DataIC50: 9.87E+3nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565487(CHEMBL4790061)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565484(CHEMBL4777518)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565492(CHEMBL4794910)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565489(CHEMBL4779788)
Affinity DataIC50: 1.06E+4nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565486(CHEMBL4789344)
Affinity DataIC50: 1.09E+4nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565493(CHEMBL4799227)
Affinity DataIC50: 1.17E+4nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565490(CHEMBL4788670)
Affinity DataIC50: 1.19E+4nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetProstaglandin G/H synthase 1(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM50565491(CHEMBL4789520)
Affinity DataIC50: 1.28E+4nMAssay Description:Inhibition of recombinant human COX1 using arachidonic acid as substrate preincubated for 5 mins followed by substrate addition and measured after 2 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetBifunctional epoxide hydrolase 2(Human)
Beni-Suef University

Curated by ChEMBL
LigandPNGBDBM11639(Celecoxib | CLX | Celebrex | 4-[5-(4-methylphenyl)...)
Affinity DataIC50: 2.61E+5nMAssay Description:Inhibition of human sEH using epoxy flour 7 as substrate measured after 30 mins by cell-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed