Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50013390
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565444BDBM50565444(CHEMBL4779776)
Affinity DataIC50: 230nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565443BDBM50565443(CHEMBL4792557)
Affinity DataIC50: 480nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565442BDBM50565442(CHEMBL4784208)
Affinity DataIC50: 930nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565442BDBM50565442(CHEMBL4784208)
Affinity DataIC50: 1.05E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565443BDBM50565443(CHEMBL4792557)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565430BDBM50565430(CHEMBL4795977)
Affinity DataIC50: 1.18E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565430BDBM50565430(CHEMBL4795977)
Affinity DataIC50: 1.31E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565435BDBM50565435(CHEMBL4787301)
Affinity DataIC50: 1.39E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565435BDBM50565435(CHEMBL4787301)
Affinity DataIC50: 1.63E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565445BDBM50565445(CHEMBL4791771)
Affinity DataIC50: 1.74E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565428BDBM50565428(CHEMBL4783925)
Affinity DataIC50: 1.74E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565431BDBM50565431(CHEMBL4792710)
Affinity DataIC50: 1.85E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565428BDBM50565428(CHEMBL4783925)
Affinity DataIC50: 2.14E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565441BDBM50565441(CHEMBL4776198)
Affinity DataIC50: 2.36E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565431BDBM50565431(CHEMBL4792710)
Affinity DataIC50: 2.46E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565441BDBM50565441(CHEMBL4776198)
Affinity DataIC50: 2.47E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565438BDBM50565438(CHEMBL4787349)
Affinity DataIC50: 2.93E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565439BDBM50565439(CHEMBL4790037)
Affinity DataIC50: 2.98E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565437BDBM50565437(CHEMBL4798678)
Affinity DataIC50: 3.15E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565439BDBM50565439(CHEMBL4790037)
Affinity DataIC50: 3.55E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565429BDBM50565429(CHEMBL4781719)
Affinity DataIC50: 3.83E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565437BDBM50565437(CHEMBL4798678)
Affinity DataIC50: 3.96E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565434BDBM50565434(CHEMBL4793354)
Affinity DataIC50: 4.05E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565438BDBM50565438(CHEMBL4787349)
Affinity DataIC50: 4.29E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565440BDBM50565440(CHEMBL4798316)
Affinity DataIC50: 4.65E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565445BDBM50565445(CHEMBL4791771)
Affinity DataIC50: 4.65E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565429BDBM50565429(CHEMBL4781719)
Affinity DataIC50: 5.45E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565444BDBM50565444(CHEMBL4779776)
Affinity DataIC50: 5.74E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565434BDBM50565434(CHEMBL4793354)
Affinity DataIC50: 5.82E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565433BDBM50565433(CHEMBL4799460)
Affinity DataIC50: 6.70E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565436BDBM50565436(CHEMBL4789799)
Affinity DataIC50: 7.03E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565436BDBM50565436(CHEMBL4789799)
Affinity DataIC50: 7.14E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565440BDBM50565440(CHEMBL4798316)
Affinity DataIC50: 8.12E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565432BDBM50565432(CHEMBL4785810)
Affinity DataIC50: 8.37E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 1(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565433BDBM50565433(CHEMBL4799460)
Affinity DataIC50: 9.03E+3nMAssay Description:Antagonist activity at human NOD1 in HEK-Blue hNOD1 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed
TargetNucleotide-binding oligomerization domain-containing protein 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565432BDBM50565432(CHEMBL4785810)
Affinity DataIC50: 9.83E+3nMAssay Description:Antagonist activity at human NOD2 in HEK-Blue hNOD2 cells assessed as secreted alkaline phosphatase reporter activity preincubated for 3 hrs followed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/30/2022
Entry Details Article
PubMed