Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50011221
TargetBeta-2 adrenergic receptor(Human)
Institute For Advanced Chemistry of Catalonia (Iqac-Csic)

Curated by ChEMBL
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataIC50: 0.480nMAssay Description:Antagonist activity at ADRB2 endogenously expressed in HEK293 cells transfected with cAMP FRET biosensor assessed as inhibition of cimaterol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Institute For Advanced Chemistry of Catalonia (Iqac-Csic)

Curated by ChEMBL
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataIC50: 0.550nMAssay Description:Antagonist activity at ADRB2 endogenously expressed in HEK293 cells transfected with cAMP FRET biosensor assessed as inhibition of cimaterol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Institute For Advanced Chemistry of Catalonia (Iqac-Csic)

Curated by ChEMBL
LigandPNGBDBM50545798(CHEMBL4633760)
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at ADRB2 endogenously expressed in HEK293 cells transfected with cAMP FRET biosensor assessed as inhibition of cimaterol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Institute For Advanced Chemistry of Catalonia (Iqac-Csic)

Curated by ChEMBL
LigandPNGBDBM50545798(CHEMBL4633760)
Affinity DataIC50: 29nMAssay Description:Antagonist activity at ADRB2 endogenously expressed in HEK293 cells transfected with cAMP FRET biosensor assessed as inhibition of cimaterol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Institute For Advanced Chemistry of Catalonia (Iqac-Csic)

Curated by ChEMBL
LigandPNGBDBM50545799(CHEMBL4634403)
Affinity DataIC50: 161nMAssay Description:Antagonist activity at ADRB2 endogenously expressed in HEK293 cells transfected with cAMP FRET biosensor assessed as inhibition of cimaterol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Institute For Advanced Chemistry of Catalonia (Iqac-Csic)

Curated by ChEMBL
LigandPNGBDBM50545799(CHEMBL4634403)
Affinity DataIC50: 594nMAssay Description:Antagonist activity at ADRB2 endogenously expressed in HEK293 cells transfected with cAMP FRET biosensor assessed as inhibition of cimaterol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Institute For Advanced Chemistry of Catalonia (Iqac-Csic)

Curated by ChEMBL
LigandPNGBDBM50545800(CHEMBL4649599)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at ADRB2 endogenously expressed in HEK293 cells transfected with cAMP FRET biosensor assessed as inhibition of cimaterol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetBeta-2 adrenergic receptor(Human)
Institute For Advanced Chemistry of Catalonia (Iqac-Csic)

Curated by ChEMBL
LigandPNGBDBM50545800(CHEMBL4649599)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at ADRB2 endogenously expressed in HEK293 cells transfected with cAMP FRET biosensor assessed as inhibition of cimaterol-induced ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed