Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50011216
TargetTumor necrosis factor(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50545753(CHEMBL4649816)
Affinity DataKd:  1.96E+4nMAssay Description:Binding affinity to recombinant TNFalpha (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as Kd for TNF-alpha-TNFR1 binding at 100 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetTumor necrosis factor(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50545753(CHEMBL4649816)
Affinity DataKd:  4.26E+3nMAssay Description:Binding affinity to recombinant TNFalpha (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as Kd for TNF-alpha-TNFR1 binding at 10 u...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetTumor necrosis factor(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50373071(CHEMBL255489)
Affinity DataKd:  9.17E+4nMAssay Description:Binding affinity to recombinant TNFalpha (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetTumor necrosis factor(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50545753(CHEMBL4649816)
Affinity DataKd:  8.21E+4nMAssay Description:Binding affinity to recombinant TNFalpha (unknown origin) expressed in Escherichia coli BL21 (DE3) incubated for 10 mins by MST assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed
TargetTumor necrosis factor(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50545753(CHEMBL4649816)
Affinity DataIC50: 109nMAssay Description:Binding affinity to recombinant TNFalpha (unknown origin) expressed in Escherichia coli BL21 (DE3) assessed as inhibition of TNFR1 binding to immobil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2021
Entry Details Article
PubMed