Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50018746
TargetProtein kinase C delta type(Human)
Ningbo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50612016BDBM50612016(CHEMBL5172923)
Affinity DataKi:  0.110nMAssay Description:Inhibition of [3H]-PDBu binding to PKCdelta C1B domain (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetProtein kinase C delta type(Human)
Ningbo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50612015BDBM50612015(CHEMBL5288713)
Affinity DataKi:  17nMAssay Description:Inhibition of [3H]-PDBu binding to PKCdelta C1B domain (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetCannabinoid receptor 1(Human)
Ningbo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50108989BDBM50108989(CHEMBL3597332)
Affinity DataKi:  470nMAssay Description:Binding affinity to human recombinant CB1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetProtein kinase C delta type(Human)
Ningbo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50612018BDBM50612018(CHEMBL5267070)
Affinity DataKi:  940nMAssay Description:Inhibition of [3H]-PDBu binding to PKCdelta C1B domain (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetProtein kinase C delta type(Human)
Ningbo University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50612017BDBM50612017(CHEMBL5284753)
Affinity DataKi:  1.40E+3nMAssay Description:Inhibition of [3H]-PDBu binding to PKCdelta C1B domain (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed