Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50013363
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 16018BDBM16018(cid_8515 | SP 600125 | ChemBiol10705 Compound 4 | ...)
Affinity DataIC50: 90nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50515263BDBM50515263(CHEMBL4531109)
Affinity DataIC50: 160nMAssay Description:Inhibition of human DDR1 using KKKSPGEYVNIEFG as substrate after 40 mins by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565131BDBM50565131(CHEMBL4795574)
Affinity DataIC50: 190nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50515263BDBM50515263(CHEMBL4531109)
Affinity DataIC50: 250nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565126BDBM50565126(CHEMBL4788894)
Affinity DataIC50: 320nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50515263BDBM50515263(CHEMBL4531109)
Affinity DataIC50: 370nMAssay Description:Inhibition of human EGFR L858R/T790M mutant GGMEDIYFEFMGGKKK as substrate measured after 40 mins in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565125BDBM50565125(CHEMBL4777530)
Affinity DataIC50: 370nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565120BDBM50565120(CHEMBL4782208)
Affinity DataIC50: 410nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565130BDBM50565130(CHEMBL4782076)
Affinity DataIC50: 430nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565128BDBM50565128(CHEMBL4800639)
Affinity DataIC50: 600nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565121BDBM50565121(CHEMBL4799531)
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565123BDBM50565123(CHEMBL4785607)
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565132BDBM50565132(CHEMBL4794035)
Affinity DataIC50: 1.68E+3nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565124BDBM50565124(CHEMBL4780101)
Affinity DataIC50: 1.75E+3nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565122BDBM50565122(CHEMBL4789089)
Affinity DataIC50: 3.48E+3nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50515263BDBM50515263(CHEMBL4531109)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of human EGFR L858R using poly[Glu:Tyr] (4:1) as substrate measured after 40 mins in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565133BDBM50565133(CHEMBL4793426)
Affinity DataIC50: 4.78E+3nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565129BDBM50565129(CHEMBL4794586)
Affinity DataIC50: 5.15E+3nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565127BDBM50565127(CHEMBL4781949)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 10(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565134BDBM50565134(CHEMBL4776996)
Affinity DataIC50: 7.37E+3nMAssay Description:Inhibition of human JNK3 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetEpithelial discoidin domain-containing receptor 1(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565131BDBM50565131(CHEMBL4795574)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human DDR1 using KKKSPGEYVNIEFG as substrate after 40 mins by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565131BDBM50565131(CHEMBL4795574)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human EGFR L858R/T790M mutant GGMEDIYFEFMGGKKK as substrate measured after 40 mins in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565131BDBM50565131(CHEMBL4795574)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human EGFR L858R using poly[Glu:Tyr] (4:1) as substrate measured after 40 mins in presence of [gamma-33P]ATP by radiometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50515263BDBM50515263(CHEMBL4531109)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK1alpha1 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 8(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565131BDBM50565131(CHEMBL4795574)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK1alpha1 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50515263BDBM50515263(CHEMBL4531109)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK2alpha2 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed
TargetMitogen-activated protein kinase 9(Human)
Peking University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50565131BDBM50565131(CHEMBL4795574)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JNK2alpha2 after 40 mins by [gamma-33ATP] radiometric assay relative to controlMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2022
Entry Details Article
PubMed