Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50010665
TargetExportin-1(Human)
Georg-August-University G£Ttingen

Curated by ChEMBL
LigandPNGBDBM50245464(CHEBI:52646 | LEPTOMYCIN B)
Affinity DataIC50: 151nMAssay Description:Inhibition of fluorescently labeled PKI phi(0)Leu NES binding to human CRM1 expressed in Escherichia coli BL21 (DE3) by fluorescence polarization com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetExportin-1(Human)
Georg-August-University G£Ttingen

Curated by ChEMBL
LigandPNGBDBM50540955(CHEMBL1450050)
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of fluorescently labeled PKI phi(0)Leu NES binding to human CRM1 expressed in Escherichia coli BL21 (DE3) by fluorescence polarization com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetExportin-1(Human)
Georg-August-University G£Ttingen

Curated by ChEMBL
LigandPNGBDBM50540956(CHEMBL4637077)
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of fluorescently labeled PKI phi(0)Leu NES binding to human CRM1 expressed in Escherichia coli BL21 (DE3) by fluorescence polarization com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetExportin-1(Human)
Georg-August-University G£Ttingen

Curated by ChEMBL
LigandPNGBDBM50540954(CHEMBL4645904)
Affinity DataIC50: 5.90E+4nMAssay Description:Inhibition of fluorescently labeled PKI phi(0)Leu NES binding to human CRM1 expressed in Escherichia coli BL21 (DE3) by fluorescence polarization com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetExportin-1(Human)
Georg-August-University G£Ttingen

Curated by ChEMBL
LigandPNGBDBM50317384(ethyl 5-(4-nitrophenyl)-4,6-dioxo-1,4,5,6-tetrahyd...)
Affinity DataIC50: 6.30E+4nMAssay Description:Inhibition of fluorescently labeled PKI phi(0)Leu NES binding to human CRM1 expressed in Escherichia coli BL21 (DE3) by fluorescence polarization com...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed