Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 50018490
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608716(CHEMBL5269322)
Affinity DataKd:  2.53E+4nMAssay Description:Binding affinity to human coagulation factor XIIIa by Spectrofluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608714(CHEMBL5281897)
Affinity DataIC50: 26nMAssay Description:Inhibition of human plasma coagulation factor XIIIa by fluorescence spectrophotometeric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608719(CHEMBL5269766)
Affinity DataIC50: 29nMAssay Description:Inhibition of human recombinant coagulation factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50164227(5-Methyl-2-(2-oxo-propylsulfanyl)-thiazolo[2,3-b][...)
Affinity DataIC50: 100nMAssay Description:Inhibition of human plasma coagulation factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608720(CHEMBL5285085)
Affinity DataIC50: 102nMAssay Description:Inhibition of human recombinant coagulation factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM577548(US11472838, Compound Ref. 22)
Affinity DataIC50: 110nMAssay Description:Inhibition of human recombinant coagulation factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608718(CHEMBL5286758)
Affinity DataIC50: 139nMAssay Description:Inhibition of human recombinant coagulation factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50136842(N-[2-(4-hydroxyphenyl)ethylacetamide | N-[2-(4-Hyd...)
Affinity DataIC50: 200nMAssay Description:Inhibition of human coagulation factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608713(CHEMBL5275210)
Affinity DataIC50: 310nMAssay Description:Inhibition of human plasma coagulation factor XIIIa by fluorescence spectrophotometeric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608710(CHEMBL5290263)
Affinity DataIC50: 350nMAssay Description:Inhibition of human plasma coagulation factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608712(CHEMBL5286863)
Affinity DataIC50: 610nMAssay Description:Inhibition of human plasma coagulation factor XIIIa by fluorescence spectrophotometeric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608711(CHEMBL5290280)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human plasma coagulation factor XIIIa by fluorescence spectrophotometeric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetProtein-glutamine gamma-glutamyltransferase 2(Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608715(CHEMBL5273935)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of tissue transglutaminase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608715(CHEMBL5273935)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of human recombinant coagulation factor XIIIa incubated for 55 mins by fluorometric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608716(CHEMBL5269322)
Affinity DataIC50: 3.62E+4nMAssay Description:Inhibition of human coagulation factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608716(CHEMBL5269322)
Affinity DataIC50: 7.63E+4nMAssay Description:Inhibition of human coagulation factor XIIIa assessed as inhibition of factor 13a mediated fibrin polymerization incubated for 24 hrs by SDS-PAGE ana...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM79403(N,N''-bis(3-azanylpropyl)butane-1,4-diamine;hydroc...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human coagulation factor XIIIa assessed as inhibition of factor 13a mediated crosslinking of fibronectin-collagen incubated for 2 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50009353(spermidine | 4-azaoctane-1,8-diamine | 4-azaoctame...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human coagulation factor XIIIa assessed as inhibition of factor 13a mediated crosslinking of fibronectin-collagen incubated for 2 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetCoagulation factor XIII A chain [Q652E](Human)
Xavier University of Louisiana

Curated by ChEMBL
LigandPNGBDBM50608717(CHEMBL5273326)
Affinity DataIC50: 1.18E+5nMAssay Description:Inhibition of human coagulation factor XIIIaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed